Antipyretics Analgesics

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Antipyretics Analgesics

Antipyretics Analgesics include NSAIDs, central analgesics, COX inhibitors, acetaminophen derivatives, and pain-relief intermediates. They represent one of the most widely used pharmaceutical categories, indicated for headaches, fever, muscle pain, joint inflammation, and viral symptoms. Their formulation versatility supports tablets, capsules, injections, and pediatric drops.

Nonsteroidal Anti-Inflammatory Drugs

Nonsteroidal anti-inflammatory drugs (NSAIDs) are widely used APIs that relieve pain, reduce fever, and suppress inflammation by inhibiting cyclooxygenase (COX) enzymes and blocking prostaglandin synthesis. NSAIDs include ibuprofen, naproxen, diclofenac, celecoxib, and many others used for musculoskeletal disorders, postoperative pain, arthritis, and acute injuries. Their pharmacological effects extend to platelet modulation and anti-thrombotic properties for certain formulations. NSAIDs are formulated into tablets, capsules, injectables, topical gels, and transdermal patches. Due to their effectiveness and broad clinical utility, NSAIDs remain foundational medications for acute and chronic inflammatory conditions, though gastrointestinal and cardiovascular risks require careful dosing.

Diclofenac Sodium CAS NO 15307-79-6

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Ibuprofen CAS NO 15687-27-1

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Ketoprofen Lysinate CAS NO 57469-78-0

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Phenylbutazone Sodium CAS NO 129-18-0

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CAS No.:129-18-0

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Oxyphenyl Butazone CAS NO 129-20-4

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Nibufin CAS NO 1224-64-2

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Ibufenac CAS NO 1553-60-2

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4,4-Diethyl-1-Phenyl-3,5-Pyrazolidinedione CAS NO 1732-61-2

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Antipyretic Analgesics

Antipyretic analgesics are APIs used to reduce fever and alleviate mild-to-moderate pain through central and peripheral mechanisms. Common agents include acetaminophen, metamizole, and combination formulations used for headaches, dental pain, musculoskeletal discomfort, and febrile illnesses. These APIs modulate prostaglandin synthesis in the central nervous system and may influence serotonergic pathways involved in pain perception. Their favorable safety profile makes them suitable for pediatric, adult, and geriatric populations. Widely formulated into tablets, syrups, suppositories, and intravenous preparations, antipyretic analgesics remain core medications in symptomatic relief and first-line therapy for nonspecific pain and fever.

Sodium Salicylate CAS NO 54-21-7

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Acetaminophen CAS NO 103-90-2

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[(2,3-Dihydro-1,5-Dimethyl-3-Oxo-2-Phenyl-1H-Pyrazol-4-Yl)Amino]Methanesulfonic Acid CAS NO 117-38-4

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2-Hydroxybenzoic Acid 4-(Acetylamino)Phenyl Ester CAS NO 118-57-0

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Acetoacet-p-Phenetidide CAS NO 122-82-7

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[(2,3-Dihydro-1,5-Dimethyl-3-Oxo-2-Phenyl-1H-Pyrazol-4-Yl)Amino]Methanesulfonic Acid Sodium Salt CAS NO 129-89-5

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2,4-Dihydro-3-Methyl-2-Phenethyl-3H-Pyrazol-3-One CAS NO 131-65-7

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Dibupyrone CAS NO 1046-17-9

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Antimigraine Drugs

Antimigraine drugs include APIs that target the neurological and vascular mechanisms underlying migraine attacks. These agents include triptans, CGRP receptor antagonists, ergot derivatives, and preventive medications such as beta-blockers and anticonvulsants. Their mechanisms involve modulation of serotonin receptors, cranial vasoconstriction, inhibition of neuropeptide release, and stabilization of neuronal excitability. Antimigraine APIs treat acute episodes and reduce attack frequency, improving quality of life for chronic sufferers. Formulations include oral tablets, nasal sprays, injectables, and fast-dissolving preparations. Their targeted pharmacological actions make antimigraine drugs central to modern headache management.

Atogepant (Mk-8031) CAS NO 1374248-81-3

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Methysergide Maleate CAS NO 129-49-7

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Cinanserin Hydrochloride CAS NO 1166-34-3

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Dihydroergotamine Mesylate CAS NO 11032-41-0

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Pizotifen CAS NO 15574-96-6

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Dehatrine CAS NO 19634-27-6

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Dihydroergocornine Tartrate CAS NO 102366-78-9

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Sumatriptan CAS NO 103628-46-2

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Antigout Drugs

Antigout drugs are APIs used to treat gout by reducing uric acid levels, controlling inflammation, and preventing acute gouty attacks. These include xanthine oxidase inhibitors such as allopurinol and febuxostat, uricosuric agents that enhance renal urate excretion, and anti-inflammatory drugs that manage painful flares. Their pharmacological actions involve inhibiting uric acid production, improving kidney clearance, and modulating inflammatory pathways activated by urate crystals. Antigout APIs are essential for long-term disease management, reduction of tophi formation, and prevention of joint damage. They are formulated into tablets, controlled-release forms, and injectables. Due to rising metabolic diseases, antigout drugs remain highly clinically relevant.

Cinchophen Hydriodide CAS NO 132-59-2

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Allopurinol CAS NO 1085-91-2

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Benzarone CAS NO 1477-19-6

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Roxburic Acid CAS NO 108657-25-6

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3,4-Dihydro-2,5,7,8-Tetramethyl-2-[2-[4-(Phenylmethyl)-1-Piperazinyl]Ethyl]-2H-1-Benzopyran-6-Ol CAS NO 114010-34-3

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Febuxostat CAS NO 144060-53-7

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n-Deacetyl-1,2,3,10-Demethyl Colchicine Hydrobromide CAS NO 152242-11-0

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(R)-Sulfinpyrazone CAS NO 159000-47-2

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Analgesics

Analgesics are APIs that provide pain relief through diverse mechanisms affecting peripheral tissues and the central nervous system. They include opioid and non-opioid agents, mixed receptor modulators, and adjuvant analgesics used for neuropathic, inflammatory, and postoperative pain. Analgesics act through pathways involving opioid receptors, prostaglandin inhibition, ion channel modulation, and neurotransmitter regulation. They are foundational in acute and chronic pain management, palliative care, and surgical recovery. Pharmaceutical forms include oral tablets, injectables, transdermal patches, suppositories, and patient-controlled analgesia systems. Their broad applicability and therapeutic importance make analgesics a cornerstone of modern medical treatment.

Ziconotide Polyacetate CAS NO 107452-89-1

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Mirogabalin Besylate CAS NO 1138245-21-2

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Triethanolamine Salicylate CAS NO 2174-16-5

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Dipipanone Hydrochloride CAS NO 125-32-6

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(+-)-Methadone Hydrochloride--Dea CAS NO 125-56-4

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R(-)-Methadone Hydrochloride Opioid Agon Ist CAS NO 125-58-6

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Trimeperidine CAS NO 125-80-4

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CAS No.:125-80-4

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Cinchophen CAS NO 132-60-5

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CAS No.:132-60-5

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