Description

Falintolol CAS NO 88134-91-2 is a selective β-adrenergic receptor antagonist (β-blocker) of significant interest in pharmaceutical research and development. Its primary value lies in its potential as a key intermediate or active pharmaceutical ingredient (API) for cardiovascular medications targeting hypertension and angina. This compound is essential for pharmaceutical manufacturers, R&D laboratories, and academic institutions engaged in the synthesis of novel therapeutic agents or generic drug development within the cardiology sector.

Application

• Pharmaceutical Intermediate: Serves as a critical building block in the multi-step synthesis of advanced β-blocker drug candidates.
• Active Pharmaceutical Ingredient (API) Research: Used in preclinical and clinical research for developing new cardiovascular therapies.
• Reference Standard: Employed as an analytical standard in quality control laboratories for method development and impurity profiling.
• Biochemical Research: Utilized in pharmacological studies to investigate β-adrenergic receptor mechanisms and selectivity.
• Generic Drug Manufacturing: A potential component in the production of generic versions of established β-blocker medications.

Basic Information

Product Name	Falintolol
CAS No.	88134-91-2
Molecular Formula	C17H27N3O4
Molecular Weight	337.42 g/mol
Synonyms	Falintolol; 1-(tert-Butylamino)-3-[(5,6,7,8-tetrahydro-6-methyl-1,8-naphthyridin-2-yl)oxy]propan-2-ol; (RS)-1-(tert-Butylamino)-3-[(5,6,7,8-tetrahydro-6-methyl-1,8-naphthyridin-2-yl)oxy]-2-propanol; BIIA 0217-CL; BIIA-0217-CL; BIIA0217CL
EINECS	Contact for details

Quality Control

Our Falintolol is manufactured under strict quality management systems. Each batch undergoes comprehensive analytical testing, including identification by spectroscopic methods (IR, NMR), purity assessment by HPLC, and control of specified impurities. A Certificate of Analysis (COA) detailing all test results is provided with every shipment to ensure traceability and compliance with your research or production standards.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at controlled room temperature (15-25°C). Due to its hygroscopic nature, the container must be kept tightly sealed in a dry environment to prevent moisture absorption. Keep away from incompatible materials.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (IR)	Conforms to reference spectrum
Identification (HPLC)	Retention time matches reference standard
Assay (HPLC)	≥ 98.0%
Related Substances (HPLC)	Total impurities ≤ 2.0% Any single unknown impurity ≤ 0.5%
Water Content (KF)	≤ 1.0%
Residue on Ignition	≤ 0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.