Description

2,3-Aziridinedicarboxylicacid,Dimethylester,(2R,3R)-(9Ci) is a high-purity, chiral aziridine derivative that serves as a critical building block in advanced organic synthesis. This compound matters for its role as a versatile intermediate in the production of complex, stereochemically defined molecules, enabling the development of novel pharmaceuticals and agrochemicals. It is primarily needed by R&D chemists and process development scientists in the pharmaceutical, biotechnology, and fine chemical industries.

Application

• Pharmaceutical Intermediate: Key chiral synthon for the synthesis of active pharmaceutical ingredients (APIs), particularly in the development of protease inhibitors, antibiotics, and other biologically active compounds.
• Agrochemical Research: Used in the creation of novel pesticides and herbicides with specific stereochemical configurations for enhanced efficacy and selectivity.
• Asymmetric Synthesis: Employed as a three-membered heterocyclic building block in ring-opening and cycloaddition reactions to introduce nitrogen and stereocenters into complex molecular architectures.
• Ligand and Catalyst Development: Serves as a precursor for the synthesis of chiral ligands and organocatalysts used in enantioselective transformations.
• Academic & Industrial R&D: Utilized in research laboratories for methodological development and the exploration of new chemical space in medicinal and synthetic chemistry.
• Fine Chemical Production: Intermediate in the multi-step synthesis of specialty chemicals requiring high enantiomeric purity.

Basic Information

Product Name	2,3-Aziridinedicarboxylicacid,Dimethylester,(2R,3R)-(9Ci)
CAS No.	154632-89-0
Molecular Formula	C7H11NO4
Molecular Weight	173.17 g/mol
Synonyms	(2R,3R)-Dimethyl Aziridine-2,3-dicarboxylate; (2R,3R)-1-Aziridine-2,3-dicarboxylic Acid Dimethyl Ester; (2R,3R)-Dimethyl 2,3-Aziridinedicarboxylate; (2R,3R)-Aziridine-2,3-dicarboxylic Acid Dimethyl Ester; (2R,3R)-Methyl Aziridine-2,3-dicarboxylate; (2R,3R)-Dimethyl cis-Aziridine-2,3-dicarboxylate; (2R,3R)-Dimethyl 1-Aziridine-2,3-dicarboxylate; (2R,3R)-1-Azabicyclo[1.1.0]butane-2,3-dicarboxylic Acid Dimethyl Ester
EINECS	Contact for details

Quality Control

Our 2,3-Aziridinedicarboxylicacid,Dimethylester,(2R,3R)-(9Ci) is produced under strict quality management protocols to ensure batch-to-batch consistency and high enantiomeric purity. Each lot undergoes comprehensive analytical testing, including chiral HPLC, to confirm identity and purity. Certificates of Analysis (COA) detailing all specifications are provided and can be tailored to meet specific customer requirements.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, well-ventilated area at a controlled room temperature (15-25°C). Keep away from heat, sparks, and open flame. This material is moisture-sensitive; keep the container tightly sealed under an inert atmosphere when not in use.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (IR)	Conforms to structure
Purity (HPLC)	≥ 98.0%
Enantiomeric Excess (Chiral HPLC)	≥ 99.0%
Melting Point	Contact for details
Loss on Drying	≤ 0.5%
Residue on Ignition	≤ 0.1%
Heavy Metals	≤ 10 ppm

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.