Description

2-[2-[2-[[6-amino-2-[1-[(2-amino-2-carbamoyl-ethyl)amino]-2-carbamoyl-ethyl]-5-methyl-pyrimidine-4-carbonyl]amino]-2-[[4-[[1-[[1-(5-amino-3,4-dihydroxy-6-methyl-oxan-2-yl)oxy-2-hydroxy-2-[4-[4-[3-(2-methyl-1-piperidyl)propylcarbamoyl]-1,3-thiazol-2-yl]-1,3-thiazol-2-yl]ethyl]carbamoyl]-2-hydroxy-propyl]carbamoyl]-3-hydroxy-butan-2-yl]carbamoyl]-1-(3H-imidazol-4-yl)ethoxy]-4,5-dihydroxy-6-(hydroxymethyl)oxan-3-yl]oxy-3,5-dihydroxy-6-(hydroxymethyl)oxan-4-yl] carbamate is a complex, high-purity synthetic intermediate of significant interest in advanced pharmaceutical research and development. This compound is valued for its intricate molecular architecture, which serves as a critical building block for novel therapeutic agents. It is primarily sought by research institutions and pharmaceutical companies engaged in the synthesis of next-generation antibiotics and other specialized bioactive molecules.

Application

• Pharmaceutical Intermediate: Serves as a key precursor in the multi-step synthesis of novel antibiotic compounds, particularly those targeting resistant bacterial strains.
• Research & Development: Used in medicinal chemistry programs for structure-activity relationship (SAR) studies and the development of new molecular entities.
• Bioconjugation Chemistry: Its functional groups make it suitable for conjugation studies in the development of antibody-drug conjugates (ADCs) or other targeted therapies.
• Enzyme Inhibition Studies: Potential application in biochemical research as a tool compound for investigating specific enzymatic pathways.
• High-Value Fine Chemical Synthesis: Employed in the production of other specialized, high-value fine chemicals and custom synthesis projects.

Basic Information

Item	Details
Product Name	2-[2-[2-[[6-amino-2-[1-[(2-amino-2-carbamoyl-ethyl)amino]-2-carbamoyl-ethyl]-5-methyl-pyrimidine-4-carbonyl]amino]-2-[[4-[[1-[[1-(5-amino-3,4-dihydroxy-6-methyl-oxan-2-yl)oxy-2-hydroxy-2-[4-[4-[3-(2-methyl-1-piperidyl)propylcarbamoyl]-1,3-thiazol-2-yl]-1,3-thiazol-2-yl]ethyl]carbamoyl]-2-hydroxy-propyl]carbamoyl]-3-hydroxy-butan-2-yl]carbamoyl]-1-(3H-imidazol-4-yl)ethoxy]-4,5-dihydroxy-6-(hydroxymethyl)oxan-3-yl]oxy-3,5-dihydroxy-6-(hydroxymethyl)oxan-4-yl] carbamate
CAS No.	77368-81-1
Molecular Formula	Contact for details
Molecular Weight	Contact for details
Synonyms	Carbamic acid, (2R,3S,4R,5R,6R)-2-[[(2R,3S,4R,5R,6R)-6-[[2-[[2-[[2-[[6-amino-2-[1-[(2-amino-2-carbamoylethyl)amino]-2-carbamoylethyl]-5-methyl-4-pyrimidinyl]carbonyl]amino]-2-[[4-[[1-[[1-(5-amino-3,4-dihydroxy-6-methyl-2-oxanyl)oxy]-2-hydroxy-2-[4-[4-[3-[(2-methyl-1-piperidinyl)propyl]carbamoyl]-2-thiazolyl]-2-thiazolyl]ethyl]carbamoyl]-2-hydroxypropyl]carbamoyl]-3-hydroxy-2-butyl]carbamoyl]-1-(1H-imidazol-4-yl)ethoxy]-4,5-dihydroxy-6-(hydroxymethyl)-3-oxanyl]oxy]-4,5-dihydroxy-2-(hydroxymethyl)oxan-3-yl] ester; Complex Macrolide/Lincosamide Intermediate; Research Code 77368-81-1.
EINECS	Contact for details

Quality Control

Our 2-[2-[2-[[6-amino-2-[1-[(2-amino-2-carbamoyl-ethyl)amino]-2-carbamoyl-ethyl]-5-methyl-pyrimidine-4-carbonyl]amino]-2-[[4-[[1-[[1-(5-amino-3,4-dihydroxy-6-methyl-oxan-2-yl)oxy-2-hydroxy-2-[4-[4-[3-(2-methyl-1-piperidyl)propylcarbamoyl]-1,3-thiazol-2-yl]-1,3-thiazol-2-yl]ethyl]carbamoyl]-2-hydroxy-propyl]carbamoyl]-3-hydroxy-butan-2-yl]carbamoyl]-1-(3H-imidazol-4-yl)ethoxy]-4,5-dihydroxy-6-(hydroxymethyl)oxan-3-yl]oxy-3,5-dihydroxy-6-(hydroxymethyl)oxan-4-yl] carbamate is manufactured under strict quality management systems. Each batch undergoes comprehensive analytical testing, including HPLC for purity and identity confirmation, to ensure it meets the stringent requirements of pharmaceutical R&D. A detailed Certificate of Analysis (COA) is provided with every shipment, documenting batch-specific results.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at a controlled room temperature (typically 15-25°C). Due to its hygroscopic nature, the container must be kept tightly sealed in a dry environment to prevent moisture uptake. For long-term storage, consider desiccants or inert atmosphere.

Specification

Item	Specification
Appearance	White to off-white solid
Identification (HPLC)	Conforms to reference standard
Identification (IR)	Conforms to structure
Assay (HPLC)	≥ 95.0%
Purity (HPLC, Area %)	≥ 97.0%
Single Unknown Impurity	≤ 1.0%
Water Content (KF)	≤ 5.0%
Residual Solvents (GC)	Complies with ICH guidelines

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.