Description

Efaroxan is a selective α-2 adrenergic receptor antagonist with significant research and pharmaceutical development applications. Its mechanism of action makes it a valuable pharmacological tool for studying autonomic nervous system functions and receptor interactions. This compound is primarily utilized by pharmaceutical R&D teams, academic researchers, and chemical manufacturers engaged in neuropharmacology and cardiovascular research.

Application

• Pharmacological Research: Used as a standard reference compound in studies investigating α-2 adrenoceptor activity and autonomic regulation.
• Neuropharmacology: A key tool for exploring central and peripheral nervous system functions, including studies on blood pressure, sedation, and analgesia.
• Drug Discovery & Development: Serves as a lead compound or intermediate in the synthesis of novel therapeutic agents targeting adrenergic pathways.
• Academic & Clinical Studies: Employed in university and institutional labs for teaching and advanced research into receptor pharmacology.
• Biochemical Assay Development: Used to validate and calibrate assays for screening potential drug candidates that interact with adrenergic receptors.
• Chemical Synthesis: Acts as a specialized intermediate for the production of more complex, receptor-targeted molecules.

Basic Information

Product Name	Efaroxan
CAS No.	89197-32-0
Molecular Formula	C13H16N2O2
Molecular Weight	232.28 g/mol
Synonyms	Efaroxan; 2-(2-Ethyl-2,3-dihydro-1,4-benzodioxin-2-yl)-4,5-dihydro-1H-imidazole; 2-(2-Ethyl-2,3-dihydro-1,4-benzodioxin-2-yl)-2-imidazoline; 2-(2-Ethyl-2,3-dihydro-1,4-benzodioxin-2-yl)-4,5-dihydro-1H-imidazole hydrochloride (common salt form); Idazoxan analog; α-2 adrenergic antagonist; Benzodioxanyl imidazoline
EINECS	Contact for details

Quality Control

Our Efaroxan is produced under strict quality management systems to ensure batch-to-batch consistency and high purity for research applications. Each lot undergoes comprehensive analytical testing, including identity confirmation, purity assay, and impurity profiling. A Certificate of Analysis (COA) detailing all test results is provided with every shipment to guarantee compliance with your research specifications.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated area at a controlled room temperature (15-25°C). Due to its hygroscopic nature, the container must be kept tightly sealed to minimize exposure to atmospheric moisture. For long-term storage, consider using desiccants.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (IR)	Conforms to structure
Purity (HPLC)	≥ 98.0%
Water Content (KF)	≤ 1.0%
Residue on Ignition	≤ 0.1%
Heavy Metals	≤ 20 ppm

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.