Description

Benzylpenicillin Diethylaminoethyl Ester Hydroiodide is a semisynthetic penicillin derivative, specifically an ester salt form designed for enhanced stability and specific pharmacological activity. This compound is critical for pharmaceutical research and development, particularly in the study of penicillin analogs and prodrug formulations. It serves as a key intermediate for researchers and manufacturers in the pharmaceutical and fine chemical sectors who require high-purity, well-characterized penicillin-based building blocks.

Application

• Pharmaceutical Intermediate: A crucial precursor in the synthesis of specialized penicillin derivatives and prodrugs for research purposes.
• Antibacterial Research: Used in microbiological and pharmacological studies to investigate structure-activity relationships (SAR) of β-lactam antibiotics.
• Reference Standard: Serves as a high-purity analytical standard for quality control and method development in pharmaceutical laboratories.
• Fine Chemical Synthesis: Employed in organic synthesis for the preparation of novel compounds with potential therapeutic applications.
• Biochemical Studies: Utilized in research exploring drug delivery mechanisms and the metabolic pathways of penicillin esters.

Basic Information

Product Name	Benzylpenicillin Diethylaminoethyl Ester Hydroiodide
CAS No.	808-71-9
Molecular Formula	C24H33IN2O4S
Molecular Weight	572.50 g/mol
Synonyms	Benzylpenicillin DEAE Ester Hydroiodide; Penicillin G Diethylaminoethyl Ester Hydroiodide; Diethylaminoethyl Ester of Benzylpenicillin Hydroiodide; 6-[(Phenylacetyl)amino]-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic Acid 2-(Diethylamino)ethyl Ester Hydroiodide; Benethamine Penicillin Iodide (related salt); DEAE-Penicillin G Hydroiodide; N,N-Diethylaminoethyl Penicillin G Hydroiodide
EINECS	Contact for details

Quality Control

Our Benzylpenicillin Diethylaminoethyl Ester Hydroiodide is produced under strict quality management systems. Each batch undergoes comprehensive analytical testing, including HPLC for purity, identity confirmation by IR and NMR spectroscopy, and tests for residual solvents and related substances. We provide full traceability and a detailed Certificate of Analysis (COA) with every shipment to ensure it meets the stringent requirements for pharmaceutical research and development.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at controlled room temperature (15-25°C). This product is hygroscopic (moisture-sensitive) and must be kept in a desiccated environment to maintain stability and purity. Keep away from incompatible materials.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (IR)	Conforms to structure
Identification (NMR)	Conforms to structure
Assay (HPLC)	≥ 98.0%
Water Content (KF)	≤ 1.0%
Related Substances (HPLC)	Total impurities ≤ 2.0%
Residual Solvents (GC)	Complies with ICH limits

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.