Description

(R)-n-Boc-2-Morpholinecarbaldehyde CAS NO 913642-85-0 is a high-purity, chiral building block of significant importance in modern organic synthesis. This compound serves as a key intermediate for the introduction of the morpholine scaffold in a stereochemically defined manner. It is primarily utilized by research chemists and process development scientists in the pharmaceutical and agrochemical industries for the synthesis of novel active ingredients and complex molecules.

Application

• Pharmaceutical Intermediate: A critical chiral precursor in the synthesis of drug candidates targeting neurological disorders, oncology, and infectious diseases.
• Agrochemical Synthesis: Used in the development of advanced pesticides and herbicides where the specific stereochemistry influences biological activity.
• Asymmetric Catalysis Ligand Synthesis: Serves as a starting material for constructing sophisticated chiral ligands and organocatalysts.
• Peptidomimetics & Bioactive Molecule Construction: Enables the incorporation of the morpholine moiety into peptide backbones and other bioactive scaffolds to modulate properties like solubility and metabolic stability.
• Academic & Process R&D: A valuable reagent for methodological development in organic chemistry and for scaling up synthetic routes under GMP-like conditions.

Basic Information

Product Name	(R)-n-Boc-2-Morpholinecarbaldehyde
CAS No.	913642-85-0
Molecular Formula	C10H17NO4
Molecular Weight	215.25 g/mol
Synonyms	(R)-tert-Butyl 2-formylmorpholine-4-carboxylate; (R)-4-(tert-Butoxycarbonyl)morpholine-2-carboxaldehyde; (R)-N-Boc-2-formylmorpholine; (R)-2-Formyl-N-Boc-morpholine; (R)-Boc-morpholine-2-carboxaldehyde; (2R)-4-[(2-Methylpropan-2-yl)oxycarbonyl]morpholine-2-carbaldehyde
EINECS	Contact for details

Quality Control

Every batch of (R)-n-Boc-2-Morpholinecarbaldehyde is manufactured and tested under strict quality management systems. We provide comprehensive analytical data to ensure the product meets the high standards required for advanced synthetic applications. A Certificate of Analysis (COA) detailing purity, chiral purity (enantiomeric excess), and impurity profile is supplied with each shipment.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at 2-8°C or as indicated on the label or COA. The product is moisture-sensitive and should be handled under inert atmosphere for long-term storage to maintain stability.

Specification

Item	Specification
Appearance	White to off-white solid
Identification (IR)	Conforms to structure
Identification (HPLC)	Conforms to reference
Purity (HPLC)	≥ 98.0%
Chiral Purity (Chiral HPLC)	≥ 99.0% ee
Water Content (KF)	≤ 0.5%
Residual Solvents (GC)	Complies with ICH guidelines

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.