Description

Aptazapine is a high-purity chemical compound of significant interest in advanced pharmaceutical research and development. Its primary value lies in its role as a key intermediate or active pharmaceutical ingredient (API) for the synthesis of novel therapeutic agents. This product is essential for R&D laboratories and manufacturers in the pharmaceutical and life sciences sectors, particularly those focused on developing new central nervous system (CNS) medications and other specialized drug candidates.

Application

• Pharmaceutical Intermediate: Serves as a critical building block in the multi-step synthesis of proprietary drug substances.
• Active Pharmaceutical Ingredient (API) Research: Used in the development and preclinical testing of new therapeutic compounds targeting specific biological pathways.
• Reference Standard: Employed as an analytical standard in quality control laboratories for method development, validation, and impurity profiling.
• Biochemical Research: Utilized in academic and industrial research to study receptor interactions, pharmacological activity, and structure-activity relationships (SAR).
• Process Development & Scale-up: Supports chemical process optimization from laboratory scale to pilot plant and commercial manufacturing.

Basic Information

Product Name	Aptazapine
CAS No.	71576-41-5
Molecular Formula	C₁₉H₂₀N₂O
Molecular Weight	292.38 g/mol
Synonyms	8-Fluoro-6-(4-methylpiperazin-1-yl)-11H-benzo[c][1]benzazepine; Aptazapinum; UNII-6V9V2RYJ6R; 6-(4-Methyl-1-piperazinyl)-8-fluoro-11H-benzo[c][1]benzazepine; 8-Fluoro-6-(4-methyl-1-piperazinyl)-11H-benzo[c][1]benzazepine
EINECS	Contact for details

Quality Control

Our Aptazapine is manufactured under strict quality management systems to ensure batch-to-batch consistency and high purity. Each lot is accompanied by a comprehensive Certificate of Analysis (COA) detailing key parameters such as identity, assay, and impurity profiles. We adhere to relevant industry standards and can support development projects requiring material suitable for use under cGMP guidelines.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, well-ventilated area at controlled room temperature (15-25°C). Due to its hygroscopic nature, the container must be kept tightly sealed to minimize exposure to atmospheric moisture. For long-term storage, consider using desiccants.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to structure
Assay (HPLC)	≥98.0%
Related Substances (HPLC)	Total impurities ≤2.0% Any single impurity ≤0.5%
Loss on Drying	≤1.0%
Residue on Ignition	≤0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.