Description

(4-((Cyclopropylamino)Methyl)-3-Fluorophenyl)Boronic Acid Hydrochloride is a high-value, functionalized boronic acid derivative designed for advanced synthetic chemistry. This compound serves as a critical building block in modern pharmaceutical and agrochemical research, enabling the formation of carbon-carbon bonds via Suzuki-Miyaura cross-coupling reactions. It is primarily sought after by R&D chemists and process development scientists in the life sciences sector for creating novel active ingredients and complex molecular architectures.

Application

• Pharmaceutical Intermediate: A key precursor in the synthesis of active pharmaceutical ingredients (APIs) for therapeutic areas such as oncology and central nervous system (CNS) disorders.
• Suzuki-Miyaura Cross-Coupling: Essential reagent for constructing biaryl and heterobiaryl scaffolds in medicinal chemistry and material science research.
• Agrochemical Research: Used in the development of novel herbicides, fungicides, and insecticides with enhanced efficacy.
• Ligand Synthesis: Building block for creating sophisticated ligands used in catalysis and metal-organic frameworks (MOFs).
• Chemical Biology Probes: Enables the synthesis of molecular probes for studying biological pathways and protein interactions.
• Material Science: Employed in the development of organic electronic materials and advanced polymers.

Basic Information

Product Name	(4-((Cyclopropylamino)Methyl)-3-Fluorophenyl)Boronic Acid Hydrochloride
CAS No.	1704096-25-2
Molecular Formula	C11H16BClFNO2
Molecular Weight	259.51 g/mol
Synonyms	(4-((Cyclopropylamino)Methyl)-3-Fluorophenyl)Boronic Acid HCl; 3-Fluoro-4-((cyclopropylamino)methyl)benzeneboronic acid hydrochloride; B-(4-((Cyclopropylamino)Methyl)-3-Fluorophenyl)boronic acid hydrochloride; (3-Fluoro-4-((cyclopropylaminomethyl)phenyl)boronic acid hydrochloride; 1704096-25-2; Boronic acid, B-[4-[(cyclopropylamino)methyl]-3-fluorophenyl]-, hydrochloride (1:1)
EINECS	Contact for details

Quality Control

Our (4-((Cyclopropylamino)Methyl)-3-Fluorophenyl)Boronic Acid Hydrochloride is manufactured under strict quality management systems to ensure batch-to-batch consistency and high purity for research and development applications. Each lot is accompanied by a comprehensive Certificate of Analysis (COA) detailing purity, identity, and impurity profiles. We support cGMP standards for advanced intermediates and can provide material suitable for non-GMP and GMP development phases upon request.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at a controlled room temperature (15-25°C). This material is hygroscopic (moisture-sensitive) and should be handled under an inert atmosphere (e.g., nitrogen or argon) when opening to prevent degradation. Keep away from incompatible materials.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to structure
Purity (HPLC)	≥ 95.0%
Water Content (KF)	≤ 2.0%
Heavy Metals	≤ 20 ppm
Residue on Ignition	≤ 0.5%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.