Description

Piboserod,2H-(1,3)Oxazino(3,2-A)Indole-10-Carboxamide, n-((1-Butyl-4-Piperidinyl)Methyl)-3,4-Dihydro- CAS NO 152811-62-6 is a high-purity, non-peptide chemical compound belonging to a class of potent and selective 5-HT4 receptor antagonists. This compound is of significant interest for its role in advanced pharmacological research and development, particularly in the study of gastrointestinal and cardiac function. It is primarily utilized by pharmaceutical R&D laboratories, contract research organizations (CROs), and academic institutions engaged in neuroscience and drug discovery programs.

Application

• Pharmaceutical Reference Standard: Serves as a certified reference material (CRM) for analytical method development, validation, and quality control in drug manufacturing.
• Mechanistic Research: Used as a selective pharmacological tool to investigate the physiological and pathophysiological roles of 5-HT4 receptors in vitro and in vivo.
• Drug Discovery & Development: Acts as a key intermediate or active pharmaceutical ingredient (API) precursor in the synthesis of novel therapeutic agents targeting serotonin-related pathways.
• Academic & Preclinical Studies: Employed in university and institutional research for studying gastrointestinal motility disorders, arrhythmias, and potential cognitive effects.
• Biochemical Assay Development: Utilized to develop and calibrate high-throughput screening (HTS) assays for receptor binding and functional activity.

Basic Information

Product Name	Piboserod,2H-(1,3)Oxazino(3,2-A)Indole-10-Carboxamide, n-((1-Butyl-4-Piperidinyl)Methyl)-3,4-Dihydro- CAS NO 152811-62-6
CAS No.	152811-62-6
Molecular Formula	C22H31N3O2
Molecular Weight	369.50 g/mol
Synonyms	Piboserod; SB-207266; SB 207266; SB207266; 2H-(1,3)Oxazino(3,2-a)indole-10-carboxamide, N-((1-butyl-4-piperidinyl)methyl)-3,4-dihydro-; N-[(1-Butylpiperidin-4-yl)methyl]-3,4-dihydro-2H-[1,3]oxazino[3,2-a]indole-10-carboxamide; 5-HT4 receptor antagonist SB-207266
EINECS	Contact for details

Quality Control

Our Piboserod is manufactured under strict quality management systems to ensure batch-to-batch consistency and high purity suitable for research applications. Each lot is accompanied by a comprehensive Certificate of Analysis (COA) detailing purity, identity, and impurity profiles. We adhere to relevant industry guidelines to support your regulatory and compliance needs.

Storage

Preserve in a tightly closed container, protected from light. Store at controlled room temperature (15-25°C) in a dry environment. For long-term storage, consider storing under inert atmosphere to maintain stability.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to reference spectrum
Identification (HPLC)	Retention time matches reference standard
Purity (HPLC)	≥98.0%
Water Content (KF)	≤0.5%
Residue on Ignition	≤0.1%
Heavy Metals	≤20 ppm

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.