Description

2-(3,4-Dihydroxy-2,5-Diaminopentanoylamino)-3-(7-Oxo-4-Oxa-1-Azabicyclo[3.2.0]Heptan-3-Yl)-3-Hydroxypropionic Acid is a complex, high-purity synthetic intermediate of significant interest in advanced pharmaceutical research and development. This compound is valued for its intricate molecular structure, which serves as a critical building block in the synthesis of novel β-lactam antibiotics and other specialized active pharmaceutical ingredients (APIs). It is primarily sought after by R&D laboratories, fine chemical manufacturers, and pharmaceutical companies engaged in the development of next-generation anti-infective therapies. Our supply ensures consistent quality and reliable availability for critical global research and production pipelines.

Application

• Pharmaceutical Intermediate: A key precursor in the synthesis of novel β-lactam antibiotic candidates and other complex therapeutic molecules.
• Research & Development: Used in medicinal chemistry for structure-activity relationship (SAR) studies and the development of new anti-infective agents.
• Fine Chemical Synthesis: Serves as a specialized building block for constructing complex heterocyclic and peptidomimetic compounds.
• API Manufacturing: Employed in the controlled, multi-step synthesis of advanced active pharmaceutical ingredients under GMP conditions where applicable.
• Biochemical Research: Potential use as a tool compound in enzymatic studies related to bacterial cell wall synthesis and inhibition.

Basic Information

Product Name	2-(3,4-Dihydroxy-2,5-Diaminopentanoylamino)-3-(7-Oxo-4-Oxa-1-Azabicyclo[3.2.0]Heptan-3-Yl)-3-Hydroxypropionic Acid
CAS No.	103059-94-5
Molecular Formula	C14H22N4O8
Molecular Weight	374.35 g/mol
Synonyms	3-(7-Oxo-4-oxa-1-azabicyclo[3.2.0]hept-3-yl)-3-hydroxy-2-[(3,4-dihydroxy-2,5-diaminopentanoyl)amino]propanoic acid; (2S,3S)-2-[[(2S,3S,4S,5R)-3,4-Dihydroxy-2,5-diaminopentanoyl]amino]-3-[(2S,5R,6R)-6-[(1R)-1-hydroxyethyl]-7-oxo-4-oxa-1-azabicyclo[3.2.0]hept-3-yl]-3-hydroxypropanoic acid (related stereoisomer); β-lactam intermediate; Advanced antibiotic synthon; Penem derivative intermediate; Carbapenem precursor analog.
EINECS	Contact for details

Quality Control

Every batch of 2-(3,4-Dihydroxy-2,5-Diaminopentanoylamino)-3-(7-Oxo-4-Oxa-1-Azabicyclo[3.2.0]Heptan-3-Yl)-3-Hydroxypropionic Acid is manufactured and analyzed under strict quality management systems. We provide comprehensive analytical documentation, including a Certificate of Analysis (COA) detailing purity, identity, and impurity profiles as determined by advanced techniques like HPLC, NMR, and mass spectrometry. Our quality commitment ensures the material meets the stringent requirements for pharmaceutical R&D and cGMP-grade synthesis upon request.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at a controlled room temperature (15-25°C). This compound is hygroscopic (moisture-sensitive); the container must be kept tightly sealed in a dry environment to prevent degradation. For long-term storage, consider desiccants or inert atmosphere.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to structure
Identification (HPLC)	Retention time matches reference standard
Assay (HPLC)	≥ 95.0%
Water Content (KF)	≤ 5.0%
Related Substances (HPLC)	Total impurities ≤ 3.0% Any single unknown impurity ≤ 1.0%
Residual Solvents (GC)	Complies with ICH guidelines

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.