Description

Fluparoxan is a selective α-2 adrenoceptor antagonist of significant interest in pharmaceutical research and development. This compound matters for its potential role in modulating neurotransmitter systems, offering a valuable tool for studying neurological pathways and developing novel therapeutic agents. It is primarily needed by research institutions, pharmaceutical companies, and contract research organizations (CROs) engaged in neuroscience, pharmacology, and central nervous system (CNS) drug discovery.

Application

• Neuroscience Research: A key pharmacological tool for investigating the function of α-2 adrenergic receptors in the brain and nervous system.
• Drug Discovery & Development: Serves as a reference standard and lead compound in the development of new CNS-targeting pharmaceuticals.
• Pharmacological Studies: Used in in vitro and in vivo assays to study receptor binding, selectivity, and signal transduction mechanisms.
• Academic Research: Employed in university and institutional labs for fundamental research into autonomic regulation and neuropsychiatric conditions.
• Biochemical Screening: Utilized in high-throughput screening (HTS) platforms to identify and characterize new chemical entities with similar activity profiles.

Basic Information

Product Name	Fluparoxan
CAS No.	101389-86-0
Molecular Formula	C15H14F3N3O
Molecular Weight	309.29 g/mol
Synonyms	Fluparoxan; 101389-86-0; 2-[2-(4-Fluorophenoxy)ethyl]-4,5-dihydro-1H-imidazole; 2-[2-(4-Fluorophenoxy)ethyl]-4,5-dihydro-1H-imidazole, monohydrochloride; BRL-44070A; BRL 44070A; BRL44070A; (RS)-Fluparoxan
EINECS	Contact for details

Quality Control

Our Fluparoxan is produced under strict quality management systems to ensure batch-to-batch consistency and reliability for research purposes. Each lot undergoes comprehensive analytical testing, including identification by spectroscopic methods (IR, NMR, MS), purity determination by HPLC, and control of related substances. A detailed Certificate of Analysis (COA) is provided with every shipment, confirming compliance with our stringent internal specifications.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at controlled room temperature (15-25°C). The product is light-sensitive and should be handled accordingly to maintain stability.

Specification

Item	Specification
Appearance	White to off-white solid
Identification (IR)	Conforms to reference spectrum
Identification (HPLC)	Retention time matches reference standard
Purity (HPLC)	≥ 98.0%
Related Substances (HPLC)	Total impurities ≤ 2.0%
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.