Description

Hymenialdisine Analogue #1 is a synthetic, small-molecule kinase inhibitor derived from the natural product hymenialdisine. This compound is of significant interest for its potent and selective inhibitory activity against key protein kinases involved in cellular signaling pathways. It serves as a critical research tool for pharmaceutical R&D, academic institutions, and biotechnology companies focused on oncology, neuroscience, and inflammatory disease research.

Application

• Biochemical Research: Used as a selective inhibitor in kinase assay development and signal transduction pathway studies.
• Pharmaceutical R&D: Serves as a lead compound or reference standard in drug discovery programs targeting cancer and neurodegenerative diseases.
• Academic Research: A key reagent for investigating the role of specific kinases in cell cycle regulation, apoptosis, and inflammation.
• Target Validation: Employed in functional genomics and proteomics to validate kinase targets in disease models.
• High-Throughput Screening (HTS): Used as a control or reference compound in screening assays to identify novel therapeutic agents.

Basic Information

Product Name	Hymenialdisine Analogue #1
CAS No.	693222-51-4
Molecular Formula	C15H12BrN5O2
Molecular Weight	374.19 g/mol
Synonyms	1H-Pyrrolo[2,3-c]azepin-8(6H)-one, 4-bromo-6-(2-hydroxyethylamino)-2-phenyl-; 4-Bromo-6-(2-hydroxyethylamino)-2-phenyl-1H-pyrrolo[2,3-c]azepin-8(6H)-one; Hymenialdisine derivative; Kinase inhibitor analogue; ALX-270-xxx (Research code series)
EINECS	Contact for details

Quality Control

Our Hymenialdisine Analogue #1 is manufactured under strict quality management systems. Each batch undergoes comprehensive analytical testing, including HPLC for purity, NMR and MS for structural confirmation, and residual solvent analysis. We provide a detailed Certificate of Analysis (COA) with every shipment, ensuring traceability and compliance with research-grade specifications. Custom synthesis and purification to meet specific project requirements are available.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at 2-8°C. This product is hygroscopic (moisture-sensitive). For long-term storage, consider desiccation or storage under an inert atmosphere. Allow the sealed vial to equilibrate to room temperature before opening to minimize moisture uptake.

Specification

Item	Specification
Appearance	Off-white to light yellow solid
Identification (HPLC)	Conforms to reference standard
Identification (NMR)	Conforms to structure
Purity (HPLC)	≥ 95.0%
Water Content (KF)	≤ 2.0%
Residual Solvents (GC)	Meets ICH guidelines

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.