Description

Pdk1-In-Rs2 CAS NO 1643958-89-7 is a potent and selective small molecule inhibitor designed to target specific kinase pathways. This compound is of significant value for biochemical and pharmacological research, enabling the study of cellular signaling mechanisms and disease pathology. It is primarily needed by researchers and developers in the pharmaceutical, biotechnology, and academic sectors for drug discovery and target validation programs.

Application

• Biochemical Research: Used as a selective tool compound to study PDK1 (3-Phosphoinositide-dependent protein kinase 1) and related signaling pathways in vitro.
• Drug Discovery & Development: Serves as a lead compound or reference standard in high-throughput screening and hit-to-lead optimization campaigns for oncology and metabolic diseases.
• Cellular Mechanism Studies: Applied in cell-based assays to investigate the role of specific kinases in cell proliferation, survival, and apoptosis.
• Target Validation: Utilized to confirm the biological and therapeutic relevance of PDK1 as a drug target in various disease models.
• Academic Research: Employed in university and institutional labs for fundamental research into kinase inhibitor structure-activity relationships (SAR).
• Preclinical Development: Acts as a pharmacological probe in animal models to assess the efficacy and pharmacokinetics of kinase inhibition.

Basic Information

Product Name	Pdk1-In-Rs2
CAS No.	1643958-89-7
Molecular Formula	Contact for details
Molecular Weight	Contact for details
Synonyms	PDK1 Inhibitor RS2; PDK1-IN-RS2; 1643958-89-7; PDK1 inhibitor; 3-Phosphoinositide-dependent protein kinase 1 inhibitor RS2; Kinase inhibitor RS2; Research compound 1643958-89-7
EINECS	Contact for details

Quality Control

Our Pdk1-In-Rs2 is produced under strict quality management protocols. Each batch undergoes rigorous analytical testing, including HPLC for purity and identity confirmation, to ensure it meets the high standards required for research applications. Certificates of Analysis (COA) with detailed chromatographic data are available upon request to support your regulatory and quality assurance needs.

Storage

Preserve in a tightly closed container, protected from light. Store at controlled room temperature (15-25°C) or as indicated on the label. This product is hygroscopic (moisture-sensitive) and must be kept in a dry environment. For long-term storage, consider desiccants or inert atmosphere.

Specification

Item	Specification
Appearance	White to off-white solid
Identification (HPLC/LC-MS)	Conforms to reference standard
Purity (HPLC)	≥ 98.0%
Water Content (KF)	≤ 1.0%
Residual Solvents (GC)	Meets ICH guidelines

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.