Description

Sstr5 Antagonist 1 is a potent and selective small molecule inhibitor targeting the somatostatin receptor subtype 5 (SSTR5). This compound is a critical research tool for investigating the role of SSTR5 in various physiological and pathological processes, including endocrine regulation and tumor biology. It is essential for pharmaceutical R&D teams, academic researchers, and biotechnology companies engaged in metabolic disorder research, neuroendocrine cancer studies, and novel therapeutic discovery programs.

Application

• Pharmacological Research: Used as a reference standard and active probe in in vitro and in vivo studies to elucidate SSTR5 signaling pathways and function.
• Drug Discovery & Development: Serves as a lead compound or molecular template for the design and optimization of new SSTR5-targeting therapeutics.
• Endocrinology Studies: Investigates the role of SSTR5 in hormone secretion, particularly insulin and glucagon, for potential applications in diabetes and metabolic syndrome research.
• Oncology Research: Explores the therapeutic potential of SSTR5 antagonism in certain neuroendocrine tumors (NETs) and other cancers where SSTR5 is expressed.
• Biochemical Assay Development: Employed as a control compound in high-throughput screening (HTS) campaigns and binding affinity assays (e.g., radioligand binding).
• Academic & Preclinical Research: Supports fundamental biological research in universities and institutes focusing on GPCR biology and receptor-specific antagonism.

Basic Information

Product Name	Sstr5 Antagonist 1
CAS No.	1628741-91-2
Molecular Formula	Contact for details
Molecular Weight	Contact for details
Synonyms	SSTR5 Antagonist-1; SSTR5 antagonist compound 1; Somatostatin Receptor 5 Antagonist 1; SSTR5 Inhibitor 1; (Research Code Compound); 1628741-91-2 (CAS Registry Number)
EINECS	Contact for details

Quality Control

Our Sstr5 Antagonist 1 is manufactured under strict quality management systems. Each batch undergoes comprehensive analytical testing, including HPLC for purity and NMR/LC-MS for structural confirmation, to ensure identity, potency, and consistency. Certificates of Analysis (COA) with detailed chromatographic data are provided to support your research integrity. We adhere to high-purity standards suitable for pharmaceutical research applications.

Storage

Preserve in a tightly closed container, protected from light. Store at -20°C or below under inert atmosphere for long-term stability. For short-term use, the product may be stored at 2-8°C. Allow the vial to equilibrate to room temperature in a desiccator before opening to prevent moisture condensation. Store in a cool, dry, and well-ventilated area away from incompatible materials.

Specification

Item	Specification
Appearance	White to off-white solid
Identification (HPLC)	Conforms to reference standard
Identification (MS)	Conforms to structure
Purity (HPLC)	≥ 98.0%
Water Content (KF)	≤ 1.0%
Residual Solvents (GC)	Complies with ICH guidelines

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.