Description

3-Fluoro-2-Morpholinopyridine-4-Boronic Acid is a high-value, multifunctional organoboron building block designed for advanced synthetic chemistry. This compound matters for its critical role as a key intermediate in cross-coupling reactions, enabling the efficient construction of complex molecular architectures. Pharmaceutical researchers and agrochemical developers need it for creating novel active ingredients, particularly in medicinal chemistry for drug discovery programs targeting a range of therapeutic areas.

Application

• Pharmaceutical Intermediate: A crucial building block in the synthesis of active pharmaceutical ingredients (APIs) for drug discovery and development.
• Suzuki-Miyaura Cross-Coupling Reactions: Serves as a versatile boronic acid reagent for forming carbon-carbon bonds to create complex biaryl and heterobiaryl structures.
• Medicinal Chemistry Research: Used in the design and synthesis of novel small molecule libraries for high-throughput screening and lead optimization.
• Agrochemical Synthesis: Employed as an intermediate in the development of new herbicides, fungicides, and insecticides.
• Material Science Precursor: Potential use in the synthesis of organic electronic materials and functional polymers.
• Contract Research & Development (CRO/CMO): Supplied to research organizations for custom synthesis and process development projects.

Basic Information

Product Name	3-Fluoro-2-Morpholinopyridine-4-Boronic Acid
CAS No.	1256355-28-8
Molecular Formula	C9H12BFN2O3
Molecular Weight	226.02 g/mol
Synonyms	3-Fluoro-2-(morpholin-4-yl)pyridine-4-boronic acid; (3-Fluoro-2-morpholinopyridin-4-yl)boronic acid; 4-Borono-3-fluoro-2-morpholinopyridine; 2-Morpholino-3-fluoropyridine-4-boronic acid; 1256355-28-8; 3-Fluoro-2-morpholin-4-ylpyridine-4-boronic acid
EINECS	Contact for details

Quality Control

Our 3-Fluoro-2-Morpholinopyridine-4-Boronic Acid is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing, including HPLC for purity and NMR for structural confirmation, to ensure it meets the high standards required for research and development. Certificates of Analysis (COA) with detailed specifications are available upon request to support your quality assurance and regulatory documentation.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at a controlled room temperature (15-25°C). Due to its hygroscopic nature, the container must be kept tightly sealed under an inert atmosphere (e.g., nitrogen or argon) to prevent moisture absorption and degradation. Keep away from incompatible materials.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to structure
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 1.0%
Heavy Metals	< 20 ppm

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.