Description

4-Fluoro-3-Iodo-5-Azaindole is a high-value halogenated azaindole derivative, a crucial building block in modern pharmaceutical and agrochemical research. Its unique molecular architecture, featuring both fluorine and iodine substituents on the azaindole core, makes it an indispensable intermediate for the synthesis of complex bioactive molecules. This compound is primarily sought after by medicinal chemists and R&D professionals in the pharmaceutical industry for developing new drug candidates, particularly in oncology and CNS therapeutic areas.

Application

• Pharmaceutical Intermediate: A key synthon for the construction of kinase inhibitors and other targeted small-molecule therapeutics.
• Agrochemical Research: Used in the development of novel herbicides and pesticides, leveraging its halogenated heterocyclic structure.
• Material Science: Serves as a precursor for advanced organic electronic materials and functional dyes.
• Chemical Biology: Employed as a probe or labeling agent in biochemical assays due to its iodine moiety.
• Academic & Contract Research: Essential for methodological development and novel synthetic route exploration in organic chemistry.

Basic Information

Product Name	4-Fluoro-3-Iodo-5-Azaindole
CAS No.	1190309-79-5
Molecular Formula	C7H4FIN2
Molecular Weight	261.93 g/mol
Synonyms	3-Iodo-4-fluoro-1H-pyrrolo[3,2-b]pyridine; 4-Fluoro-3-iodo-1H-pyrrolo[3,2-b]pyridine; 4-Fluoro-3-iodo-7-azaindole; 3-Iodo-4-fluoro-7-azaindole; 1H-Pyrrolo[3,2-b]pyridine, 4-fluoro-3-iodo-; 4-Fluoro-3-iodo-5-aza-indole
EINECS	Contact for details

Quality Control

Every batch of 4-Fluoro-3-Iodo-5-Azaindole is manufactured under strict quality management systems. Our products undergo rigorous analytical testing, including HPLC, NMR, and mass spectrometry, to ensure high purity and batch-to-batch consistency. Certificates of Analysis (COA) detailing identity, purity, and impurity profiles are provided with each shipment to support your quality assurance and regulatory needs.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at room temperature (15-25°C). This material is hygroscopic (moisture-sensitive) and light-sensitive; therefore, containers must be kept tightly sealed and stored away from direct light and moisture sources.

Specification

Item	Specification
Appearance	Off-white to light yellow crystalline powder
Identification (HPLC)	Conforms
Identification (NMR)	Conforms
Purity (HPLC)	≥97.0%
Water Content (KF)	≤0.5%
Residue on Ignition	≤0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.