Description

Apstatin Trifluoroacetate Salt CAS NO 160470-73-5 is a high-purity chemical compound primarily used as a potent and selective inhibitor of aminopeptidase P (APP). This compound is critical for biochemical research, enabling the study of peptide metabolism, inflammatory pathways, and cardiovascular functions. It is an essential tool for pharmaceutical R&D, academic institutions, and biotechnology companies focused on developing novel therapeutic agents.

Application

• Biochemical Research: A key tool for studying the role of aminopeptidase P in peptide hormone degradation and inflammatory mediator regulation.
• Pharmaceutical Development: Used in target validation and lead optimization for drug discovery programs targeting cardiovascular diseases and inflammation.
• Enzyme Inhibition Studies: Serves as a reference standard for characterizing APP enzyme kinetics and inhibition mechanisms in vitro.
• Academic Research: Employed in university and institutional labs for fundamental research into bradykinin metabolism and related physiological pathways.
• Biomarker Research: Utilized in assays to investigate APP activity as a potential biomarker in various disease states.

Basic Information

Product Name	Apstatin Trifluoroacetate Salt
CAS No.	160470-73-5
Molecular Formula	C25H38F3N5O7
Molecular Weight	577.60 g/mol
Synonyms	Apstatin TFA Salt; (2S,3R)-3-Amino-2-hydroxy-4-phenylbutanoyl-L-prolyl-L-prolyl-L-alaninamide Trifluoroacetate; Apstatin (TFA); Aminopeptidase P Inhibitor Apstatin TFA; APP Inhibitor Apstatin TFA Salt; N-[(2S,3R)-3-Amino-2-hydroxy-1-oxo-4-phenylbutyl]-L-prolyl-L-prolyl-L-alaninamide Trifluoroacetate
EINECS	Contact for details

Quality Control

Our Apstatin Trifluoroacetate Salt is manufactured under strict quality systems. Each batch undergoes comprehensive analytical testing, including HPLC for purity, NMR and MS for structural confirmation, and stringent controls for residual solvents and moisture content. Certificates of Analysis (COA) are provided, detailing all specifications and test results to ensure compliance with research-grade standards.

Storage

Preserve in a tightly closed container, protected from light. Store at -20°C or below in a freezer. This product is hygroscopic (moisture-sensitive). Allow the vial to warm to room temperature in a desiccator before opening to minimize moisture absorption.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (HPLC)	Conforms
Identification (MS)	Conforms
Purity (HPLC)	≥95.0%
Water Content (KF)	≤5.0%
Residual Solvents (GC)	Meets ICH guidelines

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.