Description

Renzapride is a selective serotonin receptor agonist with significant pharmacological activity. This compound is a critical intermediate and active pharmaceutical ingredient (API) in the research and development of novel gastrointestinal therapeutics. It is primarily utilized by pharmaceutical companies, research institutions, and contract development and manufacturing organizations (CDMOs) engaged in drug discovery and production for motility disorders.

Application

• Pharmaceutical Intermediate: Serves as a key building block in the synthesis of advanced drug candidates targeting serotonin receptors.
• Active Pharmaceutical Ingredient (API): Used in the formulation of clinical trial materials and finished dosage forms for gastrointestinal indications.
• Biomedical Research: Employed as a reference standard and tool compound in pharmacological studies to investigate 5-HT4 receptor function.
• Drug Discovery & Development: Essential for preclinical and clinical research programs focused on prokinetic agents for conditions like irritable bowel syndrome (IBS) and gastroparesis.
• Contract Manufacturing: Supplied to CDMOs for the cGMP production of bespoke pharmaceutical products under quality agreements.
• Analytical Standard: Provides a high-purity benchmark for quality control (QC) and analytical method development (e.g., HPLC, LC-MS) in laboratory settings.

Basic Information

Product Name	Renzapride
CAS No.	109872-41-5
Molecular Formula	C16H21ClN4O2
Molecular Weight	336.82 g/mol
Synonyms	Benzamide, 4-amino-5-chloro-2-methoxy-N-[(1S,4S)-5-methyl-2,5-diazabicyclo[2.2.1]hept-2-yl]-; (S)-4-Amino-5-chloro-2-methoxy-N-(1-methyl-2,5-diazabicyclo[2.2.1]hept-2-yl)benzamide; Renzapride; SB 207266 (historical); SB-207266; SB207266; Zacopride analog
EINECS	Contact for details

Quality Control

Our Renzapride is manufactured under strict quality management systems. Each batch undergoes comprehensive analytical testing to ensure identity, purity, and consistency, meeting specifications suitable for research and pharmaceutical development. A Certificate of Analysis (COA) detailing results for assay, related substances, residual solvents, and other critical parameters is provided with every shipment to ensure full traceability and compliance.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at controlled room temperature (typically 15-25°C). The product is light-sensitive and should be handled under appropriate conditions to maintain stability.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to reference spectrum
Identification (HPLC)	Retention time matches reference standard
Assay (HPLC)	≥ 98.0%
Related Substances (HPLC)	Total impurities ≤ 2.0% Any single impurity ≤ 1.0%
Loss on Drying	≤ 0.5%
Residue on Ignition	≤ 0.1%
Heavy Metals	≤ 20 ppm

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.