Description

1-[4-Methyl-2-Hexenoyl]-L-Pro-L-Leu-4,4-Dimethyl-L-Thr-2-Methyl Ala-L-Leu-L-Leu-2-Methyl Ala-2-Methyl Ala-βala-[(S)-2-(Dimethylamino)-1-Methylethyl]Nh2 is a complex, custom-designed peptide derivative that serves as a high-value intermediate or active ingredient in advanced pharmaceutical research and development. Its intricate structure, featuring multiple non-proteinogenic amino acids like 2-methylalanine and 4,4-dimethyl-L-threonine, makes it a critical tool for modulating biological activity and studying specific peptide-receptor interactions. This compound is primarily utilized by pharmaceutical companies, biotechnology research labs, and academic institutions focused on developing novel therapeutic agents, particularly in areas requiring precise molecular targeting.

Application

• Pharmaceutical Intermediate: Serves as a key building block in the synthesis of novel peptide-based drug candidates for targeted therapies.
• Biochemical Research: Used as a reference standard or probe in studies investigating enzyme inhibition, receptor binding, and signal transduction pathways.
• Drug Discovery: Employed in high-throughput screening (HTS) assays to identify and optimize lead compounds with specific biological activities.
• Peptide Mimetic Development: Acts as a core structure for creating peptidomimetics designed to enhance metabolic stability and bioavailability.
• Academic Research: Utilized in university and institutional labs for fundamental research in medicinal chemistry and peptide science.
• Contract Research & Manufacturing (CRO/CMO): Supplied to service organizations supporting the pharmaceutical industry's outsourced R&D and production needs.

Basic Information

Item	Information
Product Name	1-[4-Methyl-2-Hexenoyl]-L-Pro-L-Leu-4,4-Dimethyl-L-Thr-2-Methyl Ala-L-Leu-L-Leu-2-Methyl Ala-2-Methyl Ala-βala-[(S)-2-(Dimethylamino)-1-Methylethyl]Nh2
CAS No.	100334-46-1
Molecular Formula	C58H104N12O12
Molecular Weight	1137.5 g/mol (approx.)
Synonyms	4-Methyl-2-hexenoyl-Pro-Leu-Dmt-2-MeAla-Leu-Leu-2-MeAla-2-MeAla-β-Ala-Dma-NH2; (S)-2-(Dimethylamino)-1-methylethyl amide of 1-[4-Methyl-2-hexenoyl]-L-prolyl-L-leucyl-4,4-dimethyl-L-threonyl-2-methylalanyl-L-leucyl-L-leucyl-2-methylalanyl-2-methylalanyl-β-alanine; Custom Peptide 100334-46-1; Complex Peptide Derivative; Dmt-containing Peptide Analog; 2-MeAla Peptide
EINECS	Contact for details

Quality Control

Our 1-[4-Methyl-2-Hexenoyl]-L-Pro-L-Leu-4,4-Dimethyl-L-Thr-2-Methyl Ala-L-Leu-L-Leu-2-Methyl Ala-2-Methyl Ala-βala-[(S)-2-(Dimethylamino)-1-Methylethyl]Nh2 is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing, including HPLC for purity, MS for identity confirmation, and chiral analysis to ensure structural integrity. We provide comprehensive Certificates of Analysis (COA) with each shipment, detailing all critical quality attributes. Our production adheres to cGMP guidelines where applicable, ensuring consistency and reliability for your critical research and development projects.

Storage

Preserve in a tightly closed container, protected from light. Store at -20°C or below for long-term stability. This compound is hygroscopic (moisture-sensitive); allow the sealed vial to equilibrate to room temperature before opening to minimize moisture uptake. For extended storage, consider under an inert atmosphere such as argon or nitrogen.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (HPLC/MS)	Conforms to reference standard
Purity (HPLC)	≥ 95.0%
Single Impurity (HPLC)	≤ 1.0%
Water Content (KF)	≤ 5.0%
Peptide Content	≥ 80.0%
Specific Rotation	Contact for details

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.