Description

8-Bromo-3-Methyl-Xanthine is a high-purity, versatile xanthine derivative used as a critical intermediate in advanced organic synthesis. This compound is valued for its role in the development of pharmaceutical candidates, particularly in the research of adenosine receptor antagonists and phosphodiesterase (PDE) inhibitors. It serves the needs of research institutions, pharmaceutical R&D laboratories, and fine chemical manufacturers engaged in developing new therapeutic agents.

Application

• Pharmaceutical Intermediate: A key building block in the synthesis of novel adenosine A1 and A2A receptor antagonists for potential therapeutic applications.
• Biochemical Research: Used as a reference standard and tool compound in enzymatic studies related to PDE activity and purinergic signaling pathways.
• Medicinal Chemistry: Serves as a core scaffold for structure-activity relationship (SAR) studies to optimize drug-like properties and potency.
• Fine Chemical Synthesis: Employed in multi-step synthetic routes to create more complex heterocyclic compounds and specialized chemical entities.
• Academic Research: Utilized in university and institutional labs for fundamental research in organic chemistry and pharmacology.

Basic Information

Product Name	8-Bromo-3-Methyl-Xanthine
CAS No.	93703-24-3
Molecular Formula	C₆H₅BrN₄O₂
Molecular Weight	229.03 g/mol
Synonyms	8-Bromo-3-methyl-1H-purine-2,6-dione; 8-Bromo-3-methylxanthine; 3-Methyl-8-bromoxanthine; 8-Br-3-MX; 8-Bromo-3-methyl-3,7-dihydro-1H-purine-2,6-dione
EINECS	Contact for details

Quality Control

Our 8-Bromo-3-Methyl-Xanthine is manufactured under strict quality management systems. Each batch undergoes comprehensive analytical testing, including HPLC for purity verification and NMR/IR for structural confirmation, to ensure it meets the high standards required for research and development. A detailed Certificate of Analysis (COA) is provided with every shipment to guarantee traceability, consistency, and reliability.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at room temperature (15-25°C). The product is light-sensitive and should be handled accordingly to maintain stability.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to structure
Purity (HPLC)	≥ 98.0%
Loss on Drying	≤ 0.5%
Residue on Ignition	≤ 0.1%
Heavy Metals	≤ 20 ppm

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.