Description

2-Fluoro-3-Methoxy-Benzylamine is a versatile aromatic amine building block characterized by its unique fluorine and methoxy substituents. This compound is of significant value in advanced organic synthesis, particularly for introducing the benzylamine pharmacophore into target molecules with enhanced electronic and steric properties. It is primarily sought after by research and development teams in the pharmaceutical and agrochemical industries for the synthesis of novel active ingredients and fine chemicals.

Application

• Pharmaceutical Intermediate: A key synthon for the development of active pharmaceutical ingredients (APIs), especially in medicinal chemistry programs targeting CNS disorders, oncology, and anti-infectives.
• Agrochemical Synthesis: Used in the research and production of advanced herbicides, fungicides, and pesticides, where the fluorine atom can improve metabolic stability and bioavailability.
• Ligand and Catalyst Preparation: Serves as a precursor for chiral ligands and organocatalysts used in asymmetric synthesis.
• Material Science Research: Employed in the synthesis of specialty polymers, liquid crystals, and advanced organic electronic materials.
• Chemical Biology & Proteomics: Useful as a labeling reagent or a building block for activity-based probes and bioconjugation.
• Custom Synthesis and Contract Manufacturing: A critical starting material for custom synthesis projects and scale-up processes in fine chemical production.

Basic Information

Product Name	2-Fluoro-3-Methoxy-Benzylamine
CAS No.	93071-81-9
Molecular Formula	C8H10FNO
Molecular Weight	155.17 g/mol
Synonyms	(2-Fluoro-3-methoxyphenyl)methanamine; 1-(Aminomethyl)-2-fluoro-3-methoxybenzene; 2-Fluoro-3-methoxybenzenemethanamine; 3-Methoxy-2-fluorobenzylamine; α-Amino-2-fluoro-3-methoxytoluene; 2-Fluoro-m-anisylamine; Benzenemethanamine, 2-fluoro-3-methoxy-
EINECS	Contact for details

Quality Control

Our 2-Fluoro-3-Methoxy-Benzylamine is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing, including HPLC, GC, NMR, and MS, to ensure high purity and consistency. A comprehensive Certificate of Analysis (COA) detailing identity, purity, and impurity profiles is provided with every shipment to support your quality assurance and regulatory needs.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at room temperature (15-25°C). Due to its hygroscopic nature, the container should be kept tightly sealed under an inert atmosphere (e.g., nitrogen or argon) after opening to prevent moisture absorption and degradation.

Specification

Item	Specification
Appearance	Colorless to pale yellow liquid
Identification (IR)	Conforms to structure
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 0.5%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.