Description

5H-Imidazo(2,1-C)(1,4)Benzodiazepina is a specialized heterocyclic organic compound belonging to the benzodiazepine class, serving as a crucial advanced intermediate in modern pharmaceutical synthesis. Its fused imidazo-benzodiazepine core structure makes it a valuable building block for developing novel active pharmaceutical ingredients (APIs) with targeted therapeutic effects. This high-purity intermediate is primarily required by research institutions and pharmaceutical manufacturers engaged in the development of central nervous system (CNS) drugs, anxiolytics, and other specialty medications.

Application

• Pharmaceutical Intermediate: Key synthetic precursor in the research and production of novel benzodiazepine-derived active pharmaceutical ingredients (APIs).
• Medicinal Chemistry Research: A critical scaffold for structure-activity relationship (SAR) studies and the design of new chemical entities targeting GABA receptors.
• Preclinical Drug Development: Used in the synthesis of candidate compounds for pharmacological screening and efficacy testing.
• Contract Manufacturing: Supplied to CDMOs (Contract Development and Manufacturing Organizations) for custom synthesis projects under cGMP guidelines.
• Reference Standard: Serves as a high-purity analytical standard for quality control and regulatory submissions in pharmaceutical development.

Basic Information

Product Name	5H-Imidazo(2,1-C)(1,4)Benzodiazepina
CAS No.	78105-30-3
Molecular Formula	C₁₁H₉N₃
Molecular Weight	183.21 g/mol
Synonyms	5H-Imidazo[2,1-c][1,4]benzodiazepine; Imidazo[2,1-c][1,4]benzodiazepine; 5H-Imidazo(2,1-c)(1,4)benzodiazepine; 78105-30-3; Imidazobenzodiazepine; 5H-Imidazo(2,1-C)(1,4)Benzodiazepina [Italian]; 5H-Imidazo[2,1-c]benzodiazepine
EINECS	Contact for details

Quality Control

Our production of 5H-Imidazo(2,1-C)(1,4)Benzodiazepina adheres to stringent quality management protocols suitable for pharmaceutical intermediate applications. Each batch undergoes comprehensive analytical testing, including HPLC for purity determination and spectroscopic methods for structural confirmation. Certificates of Analysis (COA) detailing batch-specific results are provided to ensure traceability and compliance with your internal quality standards and regulatory requirements.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated area at controlled room temperature (15-25°C). Due to its hygroscopic (moisture-sensitive) nature, the container must be kept sealed under an inert atmosphere (e.g., nitrogen or argon) after opening to prevent degradation.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to structure
Purity (HPLC)	≥ 98.0%
Loss on Drying	≤ 0.5%
Residue on Ignition	≤ 0.1%
Heavy Metals	≤ 10 ppm

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.