Description

2-Fluoro-5-(4-Morpholinyl)-Benzenamine is a high-value aromatic amine derivative featuring both fluorine and morpholine substituents, making it a versatile and sought-after intermediate in advanced organic synthesis. Its molecular architecture is critical for constructing complex pharmacophores, offering unique electronic and steric properties for fine-tuning biological activity. This compound is essential for research and development chemists in the pharmaceutical and agrochemical industries, particularly for creating novel active ingredients.

Application

• Pharmaceutical Intermediate: A key building block in the synthesis of active pharmaceutical ingredients (APIs), especially for kinase inhibitors, receptor antagonists, and other small-molecule therapeutics.
• Agrochemical Research: Used in the development of new herbicides, fungicides, and insecticides, where the fluorine and morpholine groups can enhance bioavailability and target specificity.
• Material Science Precursor: Serves as a monomer or functionalization agent in the creation of specialty polymers, dyes, and advanced organic electronic materials.
• Chemical Biology Probe: Employed in the design and synthesis of molecular probes for studying enzyme mechanisms and cellular pathways.
• Custom Synthesis & Contract Manufacturing: A critical starting material for custom synthesis houses and CDMOs (Contract Development and Manufacturing Organizations) serving the global life sciences market.

Basic Information

Product Name	2-Fluoro-5-(4-Morpholinyl)-Benzenamine
CAS No.	500206-01-9
Molecular Formula	C10H13FN2O
Molecular Weight	196.22 g/mol
Synonyms	5-Amino-2-fluorophenyl morpholine; 2-Fluoro-5-morpholinoaniline; Benzenamine, 2-fluoro-5-(4-morpholinyl)-; 4-(4-Amino-3-fluorophenyl)morpholine; 3-Fluoro-6-morpholinoaniline; 2-Fluoro-5-morpholinobenzenamine; 5-Morpholino-2-fluoroaniline
EINECS	Contact for details

Quality Control

Every batch of 2-Fluoro-5-(4-Morpholinyl)-Benzenamine is manufactured and tested under a strict quality management system. We provide comprehensive analytical data to ensure the material meets the high-purity standards required for research and commercial synthesis. A detailed Certificate of Analysis (COA) is supplied with each shipment, confirming identity, purity, and impurity profiles as determined by advanced chromatographic and spectroscopic methods.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at room temperature (15-25°C). Due to its hygroscopic nature, the container must be kept tightly sealed to prevent moisture absorption, which can affect stability and performance. Keep away from incompatible materials.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (IR)	Conforms to structure
Purity (HPLC)	≥ 98.0%
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%
Single Maximum Impurity (HPLC)	≤ 0.5%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.