Description

N'-(7-[1-(2,4-Difluorophenoxy)Ethyl][1,2,4]Triazolo[1,5-A]Pyrimidin-2-Yl)-N,n-Dimethyliminoformamide is a high-purity, advanced pharmaceutical intermediate of significant commercial and research interest. This compound is valued for its role as a key building block in the synthesis of novel active pharmaceutical ingredients (APIs), particularly in therapeutic areas requiring complex heterocyclic architectures. It is primarily sought by R&D laboratories, process development chemists, and manufacturers in the global pharmaceutical and agrochemical industries for developing next-generation products.

Application

• Pharmaceutical Intermediate: Critical building block for the synthesis of novel drug candidates, especially in antiviral, antifungal, and anticancer research pipelines.
• Agrochemical Research: Used in the development of new fungicides and herbicides, leveraging the biological activity of the triazolopyrimidine core.
• Chemical Synthesis: Serves as a versatile precursor for further functionalization in medicinal chemistry and material science.
• Process Development & Scale-Up: Employed in optimizing synthetic routes from laboratory to pilot and commercial-scale production.
• Reference Standard: Used as an analytical standard for quality control and regulatory submissions in API manufacturing.
• Contract Research & Manufacturing (CRO/CMO): Supplied to organizations specializing in custom synthesis and development services.

Basic Information

Product Name	N'-(7-[1-(2,4-Difluorophenoxy)Ethyl][1,2,4]Triazolo[1,5-A]Pyrimidin-2-Yl)-N,n-Dimethyliminoformamide
CAS No.	477865-42-2
Molecular Formula	C₁₈H₁₈F₂N₆O₂
Molecular Weight	388.37 g/mol
Synonyms	N'-(7-(1-(2,4-Difluorophenoxy)ethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)-N,N-dimethylformimidamide; 477865-42-2; UNII-9J0Q8QEK0T; 9J0Q8QEK0T; N,N-Dimethyl-N'-[7-[1-(2,4-difluorophenoxy)ethyl][1,2,4]triazolo[1,5-a]pyrimidin-2-yl]formimidamide; Formimidamide, N,N-dimethyl-N'-[7-[1-(2,4-difluorophenoxy)ethyl][1,2,4]triazolo[1,5-a]pyrimidin-2-yl]-
EINECS	Contact for details

Quality Control

Our N'-(7-[1-(2,4-Difluorophenoxy)Ethyl][1,2,4]Triazolo[1,5-A]Pyrimidin-2-Yl)-N,n-Dimethyliminoformamide is manufactured under strict quality management systems. Every batch undergoes rigorous analytical testing, including HPLC, NMR, and MS, to ensure identity, purity, and consistency. We provide comprehensive Certificates of Analysis (COA) with each shipment, detailing all critical quality attributes. Our production adheres to cGMP principles where applicable, ensuring reliability for your most demanding R&D and scale-up projects.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at a controlled room temperature (15-25°C). Due to its hygroscopic (moisture-sensitive) nature, the container must be kept tightly sealed after opening to prevent degradation from atmospheric moisture. For long-term storage, consider using desiccants.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (HPLC)	Conforms to reference standard
Identification (IR)	Conforms to structure
Purity (HPLC)	≥ 98.0%
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%
Heavy Metals	≤ 10 ppm
Single Unknown Impurity (HPLC)	≤ 0.5%
Total Impurities (HPLC)	≤ 2.0%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.