Description

Deutolperisone CAS NO 474641-19-5 is a deuterated derivative of tolperisone, a centrally acting muscle relaxant. This compound is of significant interest in pharmaceutical research and development, particularly for its potential to improve the metabolic stability and pharmacokinetic profile of the parent drug. It serves as a critical intermediate or reference standard for researchers and manufacturers in the pharmaceutical industry focused on developing novel therapeutics for muscle spasticity and related neurological conditions.

Application

• Pharmaceutical Intermediate: Used in the synthesis and development of novel deuterated drug candidates, leveraging the deuterium kinetic isotope effect.
• Reference Standard: Serves as an analytical standard for quality control and method validation in pharmaceutical manufacturing and regulatory testing.
• Metabolic Studies: Employed in preclinical and clinical research to investigate the metabolic pathways and stability of tolperisone analogs.
• Active Pharmaceutical Ingredient (API) Development: A key building block for formulating new muscle relaxant medications with potentially enhanced efficacy and safety profiles.
• Isotope Labeling Research: Used in mechanistic studies and tracer experiments within medicinal chemistry and pharmacology.

Basic Information

Product Name	Deutolperisone
CAS No.	474641-19-5
Molecular Formula	C16H21D3NO
Molecular Weight	247.38 g/mol
Synonyms	2-Methyl-1-(4-methylphenyl)-3-(1-piperidinyl)-1-propanone-d3; Deuterated Tolperisone; Tolperisone-d3; 1-(4-Methylphenyl)-2-methyl-3-(piperidin-1-yl)propan-1-one-d3; (RS)-2-Methyl-1-(p-tolyl)-3-(piperidin-1-yl)propan-1-one-d3; Mydocalm-d3; Mydetone-d3
EINECS	Contact for details

Quality Control

Our Deutolperisone is manufactured under strict quality management systems. Each batch undergoes comprehensive analytical testing, including HPLC for purity and isotopic enrichment, to ensure it meets the high standards required for pharmaceutical research and development. Certificates of Analysis (COA) detailing specific batch results are available upon request.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at controlled room temperature (15-25°C). Keep the container tightly sealed in a dry environment to maintain stability.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to structure
Purity (HPLC)	≥ 98.0%
Isotopic Purity (deuterium)	≥ 98 atom % D
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.