Description

Tolperisone CAS NO 298700-23-9 is a centrally acting muscle relaxant belonging to the piperidine class of compounds. It is valued for its efficacy in reducing muscle tone and spasticity without significant sedative effects. This pharmaceutical active ingredient is primarily required by manufacturers in the pharmaceutical industry for the formulation of muscle relaxant medications.

Application

• Pharmaceutical Manufacturing: Primary active pharmaceutical ingredient (API) in prescription muscle relaxant drugs.
• Treatment of Spasticity: Formulated for conditions such as multiple sclerosis, spinal cord injuries, and other neurological disorders causing muscle stiffness.
• Muscle Pain Relief: Used in medications targeting painful muscle spasms associated with musculoskeletal conditions.
• Post-Surgical Care: Incorporated into therapeutic regimens to manage muscle rigidity following certain surgical procedures.
• Generic Drug Production: Serves as a key component for generic pharmaceutical companies producing bioequivalent versions of branded tolperisone medications.
• Clinical Research: Utilized as a reference standard or raw material in pharmacological studies and new formulation development.

Basic Information

Product Name	Tolperisone
CAS No.	298700-23-9
Molecular Formula	C16H23NO
Molecular Weight	245.36 g/mol
Synonyms	2,4'-Dimethyl-3-piperidinopropiophenone; Mydocalm; Mydetone; E-064; Caspan; Tolperisone Hydrochloride (salt form); 1-(4-Methylphenyl)-2-methyl-3-piperidin-1-ylpropan-1-one; 2-Methyl-1-(4-methylphenyl)-3-(1-piperidinyl)-1-propanone
EINECS	Contact for details

Quality Control

Our Tolperisone is manufactured under strict quality management systems. Each batch undergoes comprehensive analytical testing to ensure it meets high-purity standards suitable for pharmaceutical use. We provide full traceability and Certificates of Analysis (COA) are available for all shipments, detailing purity, identity, and impurity profiles. Our quality commitment aligns with GMP (Good Manufacturing Practice) principles and relevant ICH guidelines.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, well-ventilated place at controlled room temperature (15-25°C). Due to its hygroscopic (moisture-sensitive) nature, the container must be kept tightly sealed after opening to prevent degradation from atmospheric moisture.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (IR)	Conforms to reference spectrum
Identification (HPLC)	Retention time corresponds to reference standard
Assay (HPLC)	98.0% - 102.0% (on anhydrous basis)
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%
Related Substances (HPLC)	Individual impurity: ≤ 0.5% Total impurities: ≤ 1.5%
Heavy Metals	≤ 20 ppm

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.