Description

N2-Acetyl-D-Lysyl-L-α-Aspartyl-L-Valyl-3-Hydroxyphenylalaninamide is a synthetic peptide derivative of significant interest in advanced pharmaceutical research and development. This compound serves as a key intermediate or active pharmaceutical ingredient (API) for the development of novel therapeutic agents, particularly in areas requiring specific peptide sequences. It is primarily utilized by research institutions, pharmaceutical companies, and biotechnology firms engaged in drug discovery, process development, and the synthesis of complex bioactive molecules. The product is supplied with a focus on high purity and batch-to-batch consistency to meet stringent R&D and cGMP manufacturing requirements.

Application

• Pharmaceutical Intermediate: Serves as a critical building block in the multi-step synthesis of novel peptide-based drugs and therapeutic candidates.
• Drug Discovery Research: Used in high-throughput screening and structure-activity relationship (SAR) studies to identify and optimize new lead compounds.
• Bioconjugation & Probe Development: Acts as a substrate for developing labeled peptides, imaging agents, or targeted drug delivery systems.
• Process Chemistry & Scale-Up: Employed in the development and optimization of scalable synthetic routes for API manufacturing under cGMP conditions.
• Biochemical Research: Utilized as a tool compound to study enzyme-substrate interactions, receptor binding, or other specific biological mechanisms.
• Reference Standard: Provides a high-purity standard for analytical method development, validation, and quality control in pharmaceutical analysis.

Basic Information

Product Name	N2-Acetyl-D-Lysyl-L-α-Aspartyl-L-Valyl-3-Hydroxyphenylalaninamide
CAS No.	1239011-60-9
Molecular Formula	C31H48N6O9
Molecular Weight	648.75 g/mol
Synonyms	Ac-D-Lys-Asp-Val-3-Hydroxy-Phe-NH2; N2-Acetyl-D-lysyl-L-aspartyl-L-valyl-3-hydroxy-L-phenylalaninamide; Ac-D-Lys-L-Asp-L-Val-3-Hyp-NH2; (2S)-2-[[(2S)-2-[[(2S)-2-[[(2R)-6-acetamido-2-aminohexanoyl]amino]-3-carboxypropanoyl]amino]-3-methylbutanoyl]amino]-3-(3-hydroxyphenyl)propanamide; 3-Hydroxyphenylalanine-containing peptide derivative; CAS 1239011-60-9
EINECS	Contact for details

Quality Control

Our N2-Acetyl-D-Lysyl-L-α-Aspartyl-L-Valyl-3-Hydroxyphenylalaninamide is manufactured under strict quality systems to ensure it meets the high standards required for pharmaceutical research and development. Each batch is subjected to comprehensive analytical testing, including HPLC for purity, MS for identity confirmation, and chiral purity analysis. A detailed Certificate of Analysis (COA) is provided with each shipment, documenting the specific results for that lot. We support compliance with relevant regulatory frameworks, and custom synthesis to meet specific pharmacopeial or internal specifications is available upon request.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at a controlled room temperature (15-25°C). This product is hygroscopic (moisture-sensitive) and should be handled in a dry environment to prevent degradation. For long-term storage, consider desiccated conditions at -20°C.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (HPLC/MS)	Conforms
Purity (HPLC)	≥ 95.0%
Assay (HPLC)	≥ 98.0%
Water Content (KF)	≤ 5.0%
Heavy Metals	≤ 20 ppm
Residual Solvents (GC)	Meets ICH guidelines
Chiral Purity	≥ 99.0% ee

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.