Description

L-Arginine, N2-[[3-[(2,1,3-Benzothiadiazol-4-Ylsulfonyl)Amino]-2-Thienyl]Carbonyl]- is a specialized, high-purity synthetic derivative of the amino acid L-arginine, designed for advanced research and development applications. This compound matters for its role as a key building block or intermediate in the synthesis of novel bioactive molecules, particularly in pharmaceutical discovery. It is primarily needed by R&D chemists and process development scientists in the pharmaceutical, biotechnology, and agrochemical industries for creating new drug candidates and high-value specialty chemicals.

Application

• Pharmaceutical Intermediate: Serves as a critical synthon in the research and development of new active pharmaceutical ingredients (APIs), especially for targeted therapies.
• Bioconjugation & Probe Development: Used in the synthesis of fluorescent or affinity probes for biochemical assays and diagnostic research, leveraging the benzothiadiazole moiety.
• Peptidomimetics Research: Acts as a modified arginine residue in the design and synthesis of peptidomimetic compounds to enhance stability, bioavailability, or receptor binding.
• Chemical Biology Tool: Employed in studying enzyme-substrate interactions, signal transduction pathways, and protein-protein interactions due to its tailored functional groups.
• Agrochemical Research: Potential use as an intermediate in the development of novel crop protection agents with specific modes of action.
• Material Science Precursor: Can be utilized in the synthesis of specialized polymers or coatings with unique photophysical properties derived from its heterocyclic components.

Basic Information

Product Name	L-Arginine, N2-[[3-[(2,1,3-Benzothiadiazol-4-Ylsulfonyl)Amino]-2-Thienyl]Carbonyl]-
CAS No.	1018927-63-3
Molecular Formula	C16H18N6O5S3
Molecular Weight	486.54 g/mol
Synonyms	N2-[[3-[(2,1,3-Benzothiadiazol-4-Ylsulfonyl)Amino]-2-Thienyl]Carbonyl]-L-arginine; L-Arginine derivative with 2,1,3-benzothiadiazole-4-sulfonamide; 4-[[(3-[(2-Amino-5-guanidinopentanamido)carbonyl]-2-thienyl)amino]sulfonyl]-2,1,3-benzothiadiazole; Benzothiadiazole sulfonamide arginine derivative; BTDA-Arg; Research Compound 1018927-63-3
EINECS	Contact for details

Quality Control

Our L-Arginine derivative is produced under strict quality management protocols to ensure batch-to-batch consistency and high purity, suitable for sensitive R&D applications. Each lot undergoes comprehensive analytical characterization, including HPLC purity analysis, NMR and MS confirmation of structure, and control of specified impurities. A detailed Certificate of Analysis (COA) documenting identity, purity, and related substances is provided with every shipment to support your quality assurance and regulatory documentation needs.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at a controlled room temperature (15-25°C). The product is light-sensitive and should be handled under appropriate conditions to maintain stability. For long-term storage, consider storing under an inert atmosphere in a freezer (-20°C).

Specification

Item	Specification
Appearance	Off-white to light yellow powder
Identification (HPLC/MS)	Conforms to structure
Purity (HPLC)	≥ 95.0%
Related Substances (HPLC)	Total impurities ≤ 5.0%
Water Content (KF)	≤ 2.0%
Residual Solvents (GC)	Meets ICH guidelines

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.