Description

N2-[(Phenylmethyl)Sulfonyl]-D-Arginyl-n-[(1S)-4-[(Aminoiminomethyl)Amino]-1-Formylbutyl]Glycinamide is a high-purity, non-natural peptide derivative designed for advanced research and development applications. This compound is of significant interest due to its specific structural features, including a D-arginine residue and a formyl group, which make it a valuable building block and potential enzyme inhibitor. It is primarily utilized by pharmaceutical researchers, biotechnology companies, and academic institutions engaged in proteomics, medicinal chemistry, and biochemical pathway studies.

Application

• Pharmaceutical Research & Development: Serves as a key intermediate or reference standard in the synthesis and screening of novel therapeutic peptides and protease inhibitors.
• Biochemical Assay Development: Used as a substrate or inhibitor in enzymatic studies to investigate arginine-specific protease activity and function.
• Medicinal Chemistry: Acts as a sophisticated building block for constructing complex peptide mimetics and exploring structure-activity relationships (SAR).
• Proteomics Research: Employed in studies focusing on post-translational modifications and protein-protein interactions.
• Academic & Institutional Research: Utilized in university and government labs for fundamental research in biochemistry and molecular biology.
• Reference Standard: Provides a high-purity compound for analytical method development, validation, and quality control in GLP/GMP environments.

Basic Information

Product Name	N2-[(Phenylmethyl)Sulfonyl]-D-Arginyl-n-[(1S)-4-[(Aminoiminomethyl)Amino]-1-Formylbutyl]Glycinamide
CAS No.	186369-21-1
Molecular Formula	C₂₀H₃₄N₈O₅S
Molecular Weight	498.60 g/mol
Synonyms	D-Arg(NO2)-Gly-NH-CH(CH2CH2CH2NHC(=NH)NH2)CHO; Benzylsulfonyl-D-arginyl-glycinamide aldehyde; Bz-D-Arg-Gly-NH-CH((CH2)3NHC(=NH)NH2)CHO; Peptide aldehyde inhibitor; Protease inhibitor building block; N2-(Benzylsulfonyl)-D-arginylglycinamide, N-[(1S)-4-(aminoiminomethyl)amino-1-formylbutyl]-; (S)-N-(4-Guanidino-1-formylbutyl)-N2-(phenylmethylsulfonyl)-D-arginylglycinamide
EINECS	Contact for details

Quality Control

Our N2-[(Phenylmethyl)Sulfonyl]-D-Arginyl-n-[(1S)-4-[(Aminoiminomethyl)Amino]-1-Formylbutyl]Glycinamide is produced under strict quality management systems. Each batch undergoes comprehensive analytical testing, including HPLC for purity, MS and NMR for structural confirmation, and meets stringent in-house specifications for research-grade materials. A detailed Certificate of Analysis (COA) is provided with every shipment to ensure traceability, purity, and batch-to-batch consistency for your critical research applications.

Storage

Preserve in a tightly closed container, protected from light. Store at -20°C or below in a freezer. This product is hygroscopic (moisture-sensitive). Allow the vial to warm to room temperature in a desiccator before opening to minimize moisture absorption. For long-term storage, keep containers sealed under an inert atmosphere.

Specification

Item	Specification
Appearance	White to off-white solid
Identification (HPLC)	Conforms to reference standard
Identification (MS)	Conforms to structure
Purity (HPLC)	≥ 95.0%
Water Content (KF)	≤ 2.0%
Residual Solvents (GC)	Meets ICH guidelines

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.