Description

Bim-23127 is a high-purity, non-peptide somatostatin receptor subtype 2 (SSTR2) agonist with the CAS registry number 179188-73-9. This compound is a critical research tool for studying neuroendocrine regulation and developing targeted therapeutic strategies. It is primarily utilized by pharmaceutical R&D teams and academic researchers in the fields of endocrinology, oncology, and neuroscience for in vitro and in vivo pharmacological studies.

Application

• Pharmacological Research: Used as a selective agonist for studying somatostatin receptor subtype 2 (SSTR2) signaling pathways and functions.
• Drug Discovery & Development: Serves as a reference standard and lead compound in the development of novel therapeutics for neuroendocrine tumors (NETs) and acromegaly.
• Biochemical Assays: Employed in receptor binding studies, cAMP inhibition assays, and other in vitro screening platforms to evaluate compound efficacy and selectivity.
• Academic Research: Facilitates fundamental research into the role of somatostatin and its receptors in the central nervous system, endocrine regulation, and cell proliferation.
• Preclinical Studies: Utilized in animal models to investigate the pharmacokinetics, biodistribution, and therapeutic potential of SSTR2-targeting agents.

Basic Information

Product Name	Bim-23127
CAS No.	179188-73-9
Molecular Formula	C₂₀H₂₈N₄O₃
Molecular Weight	372.46 g/mol
Synonyms	BIM-23127; BIM 23127; (2R)-N-[(1S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-2-[[(2S)-2-Acetamidopropanoyl]amino]propanoyl]amino]-3-phenylpropan-2-yl]amino]-1-oxopropan-2-yl]carbamoyl]pyrrolidine-2-carboxamide; N-[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-2-[[(2S)-2-Acetamidopropanoyl]amino]propanoyl]amino]-3-phenylpropan-2-yl]amino]-1-oxopropan-2-yl]carbamoyl]-L-prolinamide; Somatostatin SSTR2 Agonist
EINECS	Contact for details

Quality Control

Every batch of Bim-23127 is manufactured under strict quality management systems and undergoes comprehensive analytical testing. We provide full traceability and Certificates of Analysis (COA) that detail purity, identity, and impurity profiles, ensuring compliance with research-grade standards. Our quality commitment supports reproducible and reliable results for your critical research applications.

Storage

Preserve in a tightly closed container, protected from light. Store at -20°C or below in a dry, cool place. This product is hygroscopic (moisture-sensitive). Allow the vial to equilibrate to room temperature in a desiccator before opening to minimize moisture uptake.

Specification

Item	Specification
Appearance	White to off-white solid
Identification (HPLC)	Conforms
Identification (MS)	Conforms
Purity (HPLC)	≥ 98.0%
Water Content (KF)	≤ 1.0%
Residue on Ignition	≤ 0.5%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.