Tinib Antineoplastic Drugs

Tinib Antineoplastic Drugs

Tinib antineoplastic drugs are a major class of targeted cancer therapies that inhibit dysregulated tyrosine kinases or serine/threonine kinases involved in tumor growth, angiogenesis, and metastasis. Represented by imatinib, erlotinib, gefitinib, sunitinib, sorafenib, and numerous next-generation inhibitors, these APIs block oncogenic signaling pathways such as EGFR, VEGFR, PDGFR, BCR-ABL, ALK, and RET. Their precision targeting enables high efficacy with reduced systemic toxicity compared to traditional chemotherapy. Tinib drugs are widely used in leukemia, lung cancer, renal cancer, gastrointestinal stromal tumors, and melanoma. Resistance caused by kinase mutations has led to the development of multi-targeted and mutation-specific inhibitors, making tinibs a cornerstone of precision oncology.

K-Ras(G12C) Inhibitor 6 CAS NO 2060530-16-5

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CAS No.:2060530-16-5

Grade:Pharmacy Grade

Content:99.90%

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Gdc-0077 CAS NO 2060571-02-8

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CAS No.:2060571-02-8

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Content:99.90%

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Egfr-Her2 Ex20Ins Inhibitor 1A CAS NO 2068806-31-3

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CAS No.:2068806-31-3

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Content:99.90%

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Osimertinib Dimesylate CAS NO 2070014-82-1

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CAS No.:2070014-82-1

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Content:99.90%

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Epertinib Hydrochloride CAS NO 2071195-74-7

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CAS No.:2071195-74-7

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Content:99.90%

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Jnj-64619178 CAS NO 2086772-26-9

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CAS No.:2086772-26-9

Grade:Pharmacy Grade

Content:99.90%

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Tas0728 CAS NO 2088323-16-2

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CAS No.:2088323-16-2

Grade:Pharmacy Grade

Content:99.90%

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Bi 907828 CAS NO 2095116-40-6

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CAS No.:2095116-40-6

Grade:Pharmacy Grade

Content:99.90%

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