Description

1-(3-Azetidinyl)-2-Methylpiperidine is a high-purity, advanced pharmaceutical intermediate featuring a unique fused azetidine-piperidine scaffold. This compound matters for its critical role as a sophisticated building block in modern medicinal chemistry, enabling the synthesis of complex molecules with targeted biological activity. It is primarily needed by research institutions and pharmaceutical companies engaged in the development of novel therapeutics, particularly within central nervous system (CNS) and oncology drug discovery pipelines.

Application

• Pharmaceutical Intermediate: A key chiral building block for the synthesis of novel active pharmaceutical ingredients (APIs).
• Medicinal Chemistry Research: Used in high-throughput screening and structure-activity relationship (SAR) studies to develop new drug candidates.
• Ligand Synthesis: Serves as a precursor for creating complex ligands in catalysis and receptor-binding studies.
• Chemical Biology Probes: Utilized in the development of molecular probes for studying biological pathways and enzyme functions.
• Process Chemistry Development: Employed in route scouting and optimization for scalable API manufacturing processes.

Basic Information

Product Name	1-(3-Azetidinyl)-2-Methylpiperidine
CAS No.	959239-81-7
Molecular Formula	C9H18N2
Molecular Weight	154.25 g/mol
Synonyms	2-Methyl-1-(azetidin-3-yl)piperidine; 1-(Azetidin-3-yl)-2-methylpiperidine; 2-Methyl-1-(3-azetidinyl)piperidine; Azetidine, 3-(2-methyl-1-piperidinyl)-; 3-(2-Methylpiperidin-1-yl)azetidine
EINECS	Contact for details

Quality Control

Our 1-(3-Azetidinyl)-2-Methylpiperidine is manufactured under strict quality management systems to ensure batch-to-batch consistency and high purity suitable for research and development. Each lot is accompanied by a comprehensive Certificate of Analysis (COA) detailing identity, purity, and impurity profiles. We adhere to cGMP guidelines where applicable, and our quality protocols are designed to meet the stringent requirements of pharmaceutical and advanced chemical synthesis.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at a controlled room temperature (typically 15-25°C). Due to its hygroscopic (moisture-sensitive) nature, the container must be kept tightly sealed under an inert atmosphere (e.g., nitrogen or argon) after opening to prevent degradation. Keep away from incompatible materials.

Specification

Item	Specification
Appearance	Colorless to pale yellow liquid
Identification (IR)	Conforms to structure
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.