Description

(E)-4-((6-[2-Methoxy-1-(Methoxycarbonyl)-2-Oxoethyl]-3-Pyridinyl)Amino)-4-Oxo-2-Butenoic Acid is a high-purity, non-natural amino acid derivative featuring a complex pyridine-based structure. This compound is a critical pharmaceutical intermediate and research chemical valued for its role in the synthesis of advanced bioactive molecules. It is primarily utilized by pharmaceutical R&D teams and fine chemical manufacturers developing novel therapeutic agents and chemical probes.

Application

• Pharmaceutical Intermediate: A key building block in the synthesis of complex drug candidates, particularly those targeting specific enzymatic pathways.
• Bioconjugation & Probe Development: Used to create labeled compounds and chemical probes for biochemical and cellular research due to its reactive functional groups.
• Peptidomimetic Research: Serves as a non-standard amino acid analog in the design of peptide-like molecules with enhanced stability or biological activity.
• Chemical Biology Tool: Employed in the development of activity-based probes (ABPs) and other tools for studying protein function and interaction.
• Organic Synthesis Building Block: Provides a versatile scaffold for medicinal chemists to explore new chemical space and create libraries of compounds for screening.
• Academic & Contract Research: Supplied to universities and CROs (Contract Research Organizations) for fundamental research in medicinal chemistry and drug discovery projects.

Basic Information

Item	Details
Product Name	(E)-4-((6-[2-Methoxy-1-(Methoxycarbonyl)-2-Oxoethyl]-3-Pyridinyl)Amino)-4-Oxo-2-Butenoic Acid
CAS No.	860786-07-8
Molecular Formula	C15H16N2O8
Molecular Weight	352.30 g/mol
Synonyms	4-[(6-{2-Methoxy-1-[(methoxycarbonyl)oxy]-2-oxoethyl}pyridin-3-yl)amino]-4-oxobut-2-enoic acid; (2E)-4-({6-[2-Methoxy-1-(methoxycarbonyl)-2-oxoethyl]pyridin-3-yl}amino)-4-oxo-2-butenoic Acid; 860786-07-8; 4-Oxo-2-butenoic acid, 4-((6-(2-methoxy-1-(methoxycarbonyl)-2-oxoethyl)-3-pyridinyl)amino)-, (E)-; A complex pyridine-based amino acid derivative.
EINECS	Contact for details

Quality Control

Our production of (E)-4-((6-[2-Methoxy-1-(Methoxycarbonyl)-2-Oxoethyl]-3-Pyridinyl)Amino)-4-Oxo-2-Butenoic Acid adheres to stringent quality management protocols. Every batch undergoes comprehensive analytical testing, including HPLC for purity and NMR/LC-MS for structural confirmation, to ensure it meets the exacting standards required for pharmaceutical research. A detailed Certificate of Analysis (COA) is provided with each shipment, documenting purity, identity, and impurity profiles.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at a controlled room temperature (15-25°C). This compound is hygroscopic (moisture-sensitive); the container must be kept tightly sealed in a dry environment to prevent degradation. For long-term storage, consider storage under an inert atmosphere.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to structure
Identification (HPLC)	Retention time matches reference standard
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 1.0%
Residue on Ignition	≤ 0.5%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.