Description

2-Azetidinecarboxamide,3-Amino-n-Methyl-4-Oxo-,cis-(9Ci) is a high-purity, specialized heterocyclic organic compound featuring a cis-configured azetidine ring. This molecule is valued for its role as a critical chiral building block and intermediate in advanced synthetic chemistry. It is primarily sought after by research institutions and pharmaceutical companies engaged in the development of novel active pharmaceutical ingredients (APIs), peptidomimetics, and other fine chemicals where stereochemical control is paramount.

Application

• Pharmaceutical Intermediate: Serves as a key chiral synthon in the research and synthesis of novel drug candidates, particularly in oncology and central nervous system (CNS) therapeutic areas.
• Peptidomimetics Research: Used to construct constrained scaffolds that mimic peptide structures, enhancing metabolic stability and bioavailability in drug design.
• Asymmetric Synthesis: Employed as a building block in catalytic asymmetric reactions to introduce the azetidine moiety with high enantiomeric purity.
• Chemical Biology Probes: Utilized in the development of molecular probes and tool compounds for studying enzyme mechanisms and protein-ligand interactions.
• Agrochemical Research: Investigated as an intermediate for creating new generations of herbicides or fungicides with novel modes of action.
• Material Science: Potential use in the synthesis of specialized polymers or ligands for catalysis.

Basic Information

Product Name	2-Azetidinecarboxamide,3-Amino-n-Methyl-4-Oxo-,cis-(9Ci)
CAS No.	84209-05-2
Molecular Formula	C5H9N3O2
Molecular Weight	143.15 g/mol
Synonyms	cis-3-Amino-N-methyl-4-oxoazetidine-2-carboxamide; (2R,3S)-3-Amino-N-methyl-4-oxoazetidine-2-carboxamide; 3-Amino-N-methyl-4-oxo-2-azetidinecarboxamide, cis-; 2-Azetidinecarboxamide, 3-amino-N-methyl-4-oxo-, (2R,3S)-; Azetidine-2-carboxamide, 3-amino-N-methyl-4-oxo-, cis-; A building block for β-lactam analogs.
EINECS	Contact for details

Quality Control

Every batch of our 2-Azetidinecarboxamide,3-Amino-n-Methyl-4-Oxo-,cis-(9Ci) is manufactured under strict quality management systems. We provide comprehensive analytical documentation, including Certificates of Analysis (COA) detailing purity, chiral purity, and impurity profiles as determined by advanced techniques like HPLC and NMR. Our quality commitment ensures material suitable for demanding GMP-grade pharmaceutical R&D applications.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at a controlled room temperature (15-25°C). Due to its hygroscopic (moisture-sensitive) nature, the container must be kept tightly sealed in a dry environment to prevent degradation. For long-term storage, consider using desiccants.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (IR)	Conforms to structure
Purity (HPLC)	≥ 98.0%
Chiral Purity (Chiral HPLC)	≥ 99.0% ee
Water Content (KF)	≤ 1.0%
Residue on Ignition	≤ 0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.