Description

Bifeprunox Mesylate is a high-purity pharmaceutical intermediate and research chemical. This compound is significant for its role in the development of novel antipsychotic agents targeting dopamine and serotonin receptors. It is primarily required by pharmaceutical R&D laboratories, API manufacturers, and academic institutions engaged in neuropharmacology and central nervous system (CNS) drug discovery.

Application

• Pharmaceutical Intermediate: Key building block in the synthesis of advanced antipsychotic drug candidates.
• Research & Development: Used as a reference standard and active compound in preclinical studies for neurological disorders.
• Mechanistic Studies: Employed in biochemical assays to investigate dopamine D2 and serotonin 5-HT1A receptor partial agonism.
• API Manufacturing: Serves as a critical starting material or intermediate in the production of active pharmaceutical ingredients (APIs).
• Academic Research: Utilized in university and institutional labs for neuroscience and psychopharmacology research projects.
• Process Chemistry: Applied in route scouting and optimization for the scalable synthesis of related therapeutic compounds.

Basic Information

Product Name	Bifeprunox Mesylate
CAS No.	350992-13-1
Molecular Formula	C₂₄H₂₉N₃O₃ • CH₄O₃S
Molecular Weight	503.58 g/mol
Synonyms	7-[4-([1,1'-Biphenyl]-3-ylmethyl)piperazin-1-yl]-1,3-benzoxazol-2(3H)-one methanesulfonate; DU-127090; Bifeprunox methanesulfonate; UNII-6V8V8TPN8W
EINECS	Contact for details

Quality Control

Our Bifeprunox Mesylate is manufactured under strict quality management systems. Each batch undergoes comprehensive analytical testing, including HPLC for purity, residual solvent analysis, and identity confirmation (IR, NMR) to ensure it meets the stringent requirements for pharmaceutical research and development. Certificates of Analysis (COA) with detailed chromatographic data are provided to guarantee traceability and batch-to-batch consistency.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at controlled room temperature (15-25°C). Due to its hygroscopic (moisture-sensitive) nature, the container must be kept tightly sealed in a dry environment to prevent degradation.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to structure
Identification (HPLC)	Retention time matches reference
Assay (HPLC)	≥98.0%
Related Substances (HPLC)	Total impurities ≤2.0%
Water Content (KF)	≤1.0%
Residual Solvents (GC)	Complies with ICH limits

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.