Description

(+/-)-Ethylketazocine CAS NO 36292-66-7 is a synthetic opioid receptor ligand of significant interest in pharmacological research. This compound is valued for its role as a potent and selective κ-opioid receptor agonist, making it a critical tool for studying receptor function and signal transduction pathways. It is primarily utilized by pharmaceutical R&D teams, academic research institutions, and contract research organizations (CROs) focused on neuroscience, pain management, and neuropharmacology.

Application

• Neuroscience Research: A key pharmacological tool for investigating the function and distribution of κ-opioid receptors (KOR) in the central nervous system.
• Analgesic Studies: Used in preclinical models to study κ-opioid mediated analgesia and to understand mechanisms of pain modulation.
• Receptor Binding Assays: Serves as a standard or reference compound in competitive binding experiments to characterize new chemical entities.
• Signal Transduction Research: Employed to study downstream effects of KOR activation, including G-protein coupling and second messenger systems.
• Behavioral Pharmacology: Utilized in animal studies to explore the effects of κ-opioid activation on behavior, mood, and stress responses.
• Drug Discovery & Development: Acts as a benchmark compound for the screening and validation of novel analgesic and psychotherapeutic candidates.

Basic Information

Product Name	(+/-)-Ethylketazocine
CAS No.	36292-66-7
Molecular Formula	C19H27NO
Molecular Weight	285.43 g/mol
Synonyms	Ethylketazocine; Win 35,197-2; (±)-Ethylketazocine; Ethylketocyclazocine; 2-(3,4-Dichlorophenyl)-N-methyl-N-[(1S,2S)-2-pyrrolidin-1-ylcyclohexyl]acetamide (non-specific isomer); U-50488 (related analog); Ketazocine analog; Kappa opioid agonist EKC
EINECS	Contact for details

Quality Control

Our (+/-)-Ethylketazocine is produced and handled under strict quality management protocols to ensure batch-to-batch consistency and reliability for research applications. Each lot undergoes comprehensive analytical testing, including identity confirmation by spectroscopic methods and purity assessment by HPLC. A Certificate of Analysis (COA) detailing specific results is provided with every shipment to support your regulatory and documentation requirements.

Storage

Preserve in a tightly closed container, protected from light. Store at controlled room temperature (15-25°C) in a dry, well-ventilated area. Keep the container sealed to protect this light-sensitive material from degradation.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to reference spectrum
Identification (HPLC)	Retention time matches reference standard
Purity (HPLC)	≥ 98.0%
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%
Heavy Metals	≤ 20 ppm

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.