Description

4-Fluoro-2-(Morpholinomethyl)Phenylboronic Acid Pinacol Ester is a sophisticated boronic ester derivative designed for advanced synthetic chemistry. This compound matters as a key protected boronic acid building block, offering enhanced stability and solubility for complex coupling reactions. Pharmaceutical researchers and fine chemical manufacturers need it for the development of novel active pharmaceutical ingredients (APIs) and other high-value organic molecules through Suzuki-Miyaura cross-coupling.

Application

• Pharmaceutical Intermediate Synthesis: A crucial building block for constructing complex molecules in API research and development.
• Suzuki-Miyaura Cross-Coupling Reactions: Serves as a stable, protected boronic acid reagent for forming carbon-carbon bonds in complex organic synthesis.
• Ligand and Catalyst Development: Used in the preparation of novel ligands and organometallic catalysts for asymmetric synthesis.
• Material Science Research: Employed in the synthesis of organic electronic materials and advanced polymers.
• Agrochemical Intermediate Production: A key precursor in the synthesis of novel herbicides and fungicides.
• Academic and R&D Laboratories: Essential for methodological studies and exploratory chemistry in academic and industrial settings.

Basic Information

Product Name	4-Fluoro-2-(Morpholinomethyl)Phenylboronic Acid Pinacol Ester
CAS No.	2096340-33-7
Molecular Formula	C₁₇H₂₅BFNO₃
Molecular Weight	321.20 g/mol
Synonyms	2-(4-Fluoro-2-(morpholinomethyl)phenyl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane; 4-Fluoro-2-(morpholin-4-ylmethyl)phenylboronic acid pinacol ester; (4-Fluoro-2-((morpholin-4-yl)methyl)phenyl)boronic acid pinacol ester; 4,4,5,5-Tetramethyl-2-[4-fluoro-2-(morpholinomethyl)phenyl]-1,3,2-dioxaborolane; B-[4-Fluoro-2-[(4-morpholinyl)methyl]phenyl]-4,4,5,5-tetramethyl-1,3,2-dioxaborolane; CAS 2096340-33-7; 4-Fluoro-2-morpholinomethylphenylboronic acid pinacol ester.
EINECS	Contact for details

Quality Control

Our 4-Fluoro-2-(Morpholinomethyl)Phenylboronic Acid Pinacol Ester is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing, including HPLC, NMR, and LC-MS, to ensure high purity and batch-to-batch consistency. Certificates of Analysis (COA) detailing identity, purity, and impurity profiles are available upon request to support your quality assurance and regulatory documentation needs.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at a controlled room temperature (15-25°C). Due to its hygroscopic nature, the container must be kept tightly sealed in a dry environment to prevent moisture absorption, which can affect stability and performance.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (HPLC)	Conforms
Identification (NMR)	Conforms
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.