Description

Boronic Acid, B-[4-(1-Piperidinylsulfonyl)-2-(Trifluoromethyl)Phenyl]- is a high-value, functionalized arylboronic acid derivative designed for advanced synthetic applications. This compound is a critical building block in modern pharmaceutical and agrochemical research, enabling the formation of carbon-carbon bonds via the versatile Suzuki-Miyaura cross-coupling reaction. It is primarily sought after by R&D chemists and process development scientists in the life sciences sector for the synthesis of complex molecules targeting a range of therapeutic areas.

Application

• Pharmaceutical Intermediate: A key precursor in the synthesis of active pharmaceutical ingredients (APIs), particularly for candidates containing trifluoromethyl and sulfonamide pharmacophores.
• Agrochemical Research: Used in the development of novel herbicides, fungicides, and insecticides, leveraging its unique structural motifs for bioactivity.
• Material Science: Serves as a monomer or functionalization agent in the creation of advanced polymers and organic electronic materials.
• Suzuki-Miyaura Cross-Coupling: An essential reagent for palladium-catalyzed coupling reactions to construct biaryl and heterobiaryl structures central to medicinal chemistry.
• Chemical Biology & Proteomics: Utilized as a handle for bioconjugation and the development of chemical probes and inhibitors.
• Catalyst Ligand Synthesis: Acts as a precursor for synthesizing specialized ligands used in homogeneous catalysis.

Basic Information

Product Name	Boronic Acid, B-[4-(1-Piperidinylsulfonyl)-2-(Trifluoromethyl)Phenyl]-
CAS No.	2096339-82-9
Molecular Formula	C12H15BF3NO4S
Molecular Weight	337.12 g/mol
Synonyms	[4-(Piperidine-1-sulfonyl)-2-(trifluoromethyl)phenyl]boronic acid; 2-(Trifluoromethyl)-4-(1-piperidinylsulfonyl)benzeneboronic acid; 4-(1-Piperidinosulfonyl)-2-(trifluoromethyl)phenylboronic acid; B-[4-(Piperidin-1-ylsulfonyl)-2-(trifluoromethyl)phenyl]boronic acid; (4-(Piperidine-1-sulfonyl)-2-(trifluoromethyl)phenyl)boronic acid
EINECS	Contact for details

Quality Control

Our Boronic Acid, B-[4-(1-Piperidinylsulfonyl)-2-(trifluoromethyl)Phenyl]- is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing, including HPLC, NMR, and elemental analysis, to ensure high purity and batch-to-batch consistency. Certificates of Analysis (COA) detailing identity, purity, and impurity profiles are available upon request. We support development and production needs from milligram to kilogram scale with reliable quality.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at a controlled room temperature (15-25°C). This material is hygroscopic (moisture-sensitive) and easily oxidized; for long-term storage, it is recommended to keep the container under an inert atmosphere (e.g., nitrogen or argon) in a desiccator.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (IR)	Conforms to structure
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 0.5%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.