Description

(2-Fluoro-4-Methyl-5-(Morpholinosulfonyl)Phenyl)Boronic Acid is a sophisticated arylboronic acid derivative designed for advanced cross-coupling reactions. This compound matters as a key building block in modern pharmaceutical and agrochemical research, enabling the precise construction of complex molecules. It is primarily needed by R&D chemists and process development scientists in the pharmaceutical, agrochemical, and material science industries for synthesizing novel active ingredients and functional materials.

Application

• Pharmaceutical Intermediate: A critical precursor in Suzuki-Miyaura cross-coupling reactions for synthesizing novel drug candidates, particularly in kinase inhibitor and oncology research.
• Agrochemical Synthesis: Used to create advanced active ingredients for crop protection products, leveraging the fluorine and sulfonyl substituents for enhanced bioactivity and stability.
• Material Science Research: Serves as a monomer or functionalization agent in the development of organic electronic materials, such as polymers for OLEDs and sensors.
• Chemical Biology Probes: Employed in the synthesis of bioconjugates and molecular probes for studying biological pathways and target engagement.
• Process Chemistry & Scale-up: Utilized in route development and optimization for the commercial-scale production of fine chemicals and APIs.
• Custom Synthesis & Contract Manufacturing: A valuable starting material for CROs and CDMOs offering bespoke chemical synthesis services to global clients.

Basic Information

Product Name	(2-Fluoro-4-Methyl-5-(Morpholinosulfonyl)Phenyl)Boronic Acid
CAS No.	1704121-24-3
Molecular Formula	C11H15BFNO4S
Molecular Weight	287.12 g/mol
Synonyms	5-(Morpholinosulfonyl)-2-fluoro-4-methylbenzeneboronic acid; [2-Fluoro-4-methyl-5-(4-morpholinosulfonyl)phenyl]boronic acid; 2-Fluoro-4-methyl-5-morpholinosulfonylphenylboronic acid; Boronic acid, B-[2-fluoro-4-methyl-5-[(4-morpholinyl)sulfonyl]phenyl]-; 1704121-24-3; (2-Fluoro-4-methyl-5-(morpholine-4-sulfonyl)phenyl)boronic acid
EINECS	Contact for details

Quality Control

Our (2-Fluoro-4-Methyl-5-(Morpholinosulfonyl)Phenyl)Boronic Acid is manufactured under strict quality management systems. Every batch undergoes rigorous analytical testing, including HPLC, NMR, and elemental analysis, to ensure high purity and batch-to-batch consistency. Certificates of Analysis (COA) detailing all specifications are provided and available upon request to support your quality assurance and regulatory documentation needs.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at a controlled room temperature (15-25°C). Due to its hygroscopic (moisture-sensitive) nature, the container must be kept tightly sealed under an inert atmosphere (e.g., nitrogen or argon) after opening to prevent degradation.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (IR)	Conforms to structure
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 1.0%
Heavy Metals	≤ 20 ppm
Residue on Ignition	≤ 0.5%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.