Description

(2-Fluoro-5-(((4-Methoxybenzyl)Amino)Methyl)Phenyl)Boronic Acid is a sophisticated boronic acid derivative featuring a fluorinated aromatic core and a methoxybenzyl-protected amino linker. This compound matters as a high-value building block in modern synthetic chemistry, enabling the precise construction of complex molecules through robust cross-coupling reactions. It is primarily needed by research and development teams in the pharmaceutical and agrochemical industries for creating novel active ingredients and advanced materials.

Application

• Pharmaceutical Intermediate: A key precursor in Suzuki-Miyaura cross-coupling reactions for synthesizing novel drug candidates, particularly in oncology and CNS therapeutic areas.
• Agrochemical Research: Used to construct complex molecular scaffolds for developing new-generation pesticides and herbicides with improved efficacy.
• Material Science: Serves as a monomer or functionalization agent in the synthesis of advanced polymers, OLED materials, and liquid crystals.
• Chemical Biology & Proteomics: Employed as a handle for bioconjugation and the development of activity-based probes and sensors.
• Academic & Contract Research: Essential for methodological development in organic synthesis and catalysis research within university and CRO laboratories.
• Library Synthesis: Used by medicinal chemistry groups for the parallel synthesis of diverse compound libraries to explore structure-activity relationships (SAR).

Basic Information

Item	Detail
Product Name	(2-Fluoro-5-(((4-Methoxybenzyl)Amino)Methyl)Phenyl)Boronic Acid
CAS No.	1704121-17-4
Molecular Formula	C15H17BFNO3
Molecular Weight	289.11 g/mol
Synonyms	5-[(4-Methoxybenzylamino)methyl]-2-fluorophenylboronic acid; 2-Fluoro-5-[[(4-methoxyphenyl)methylamino]methyl]benzeneboronic acid; [2-Fluoro-5-[[(4-methoxyphenyl)methylamino]methyl]phenyl]boronic acid; Boronic acid, B-[2-fluoro-5-[[[(4-methoxyphenyl)methyl]amino]methyl]phenyl]-; 1704121-17-4; AKOS026712293; FT-0773297
EINECS	Contact for details

Quality Control

Our (2-Fluoro-5-(((4-Methoxybenzyl)Amino)Methyl)Phenyl)Boronic Acid is manufactured under strict quality management systems. Every batch undergoes comprehensive analytical characterization including HPLC, NMR, and MS to confirm identity and purity. We provide a detailed Certificate of Analysis (COA) with each shipment, ensuring full traceability and compliance with your research or production specifications.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at a controlled room temperature (15-25°C). Due to its hygroscopic nature, the container must be kept tightly sealed in a dry environment to prevent moisture absorption and potential decomposition. For long-term storage, consider using desiccants or an inert atmosphere.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to structure
Identification (NMR)	Conforms to structure
Purity (HPLC)	≥ 95%
Water Content (KF)	≤ 1.0%
Heavy Metals	≤ 20 ppm

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.