Description

(2-Fluoro-5-((4-Methylpiperidin-1-yl)sulfonyl)phenyl)boronic acid is a high-value, synthetically versatile organoboron building block. This compound is critical for modern pharmaceutical and agrochemical research, enabling the efficient construction of complex molecules through cross-coupling reactions. It is primarily needed by R&D chemists and process development scientists in the pharmaceutical, agrochemical, and advanced materials industries for creating novel active ingredients and functional molecules.

Application

• Pharmaceutical Intermediate: A key reagent in Suzuki-Miyaura cross-coupling reactions for synthesizing novel drug candidates, particularly in kinase inhibitor and CNS-targeted therapeutic research.
• Agrochemical Development: Used to construct complex heterocyclic scaffolds for next-generation herbicides, fungicides, and insecticides with improved efficacy and environmental profiles.
• Material Science Research: Serves as a precursor for creating functionalized polymers, liquid crystals, and organic electronic materials via its boronic acid functionality.
• Chemical Biology & Probe Synthesis: Employed in the synthesis of molecular probes and bioconjugates for studying biological pathways and protein interactions.
• Process Chemistry & Scale-up: Provides a reliable and scalable building block for optimizing synthetic routes from laboratory to pilot plant scale.
• Contract Research & Manufacturing (CRO/CMO): Supplied to service organizations that require high-purity, specialized boronates for client-directed synthesis projects.

Basic Information

Item	Details
Product Name	(2-Fluoro-5-((4-Methylpiperidin-1-yl)sulfonyl)phenyl)boronic Acid
CAS No.	1704097-14-2
Molecular Formula	C12H17BFNO4S
Molecular Weight	301.15 g/mol
Synonyms	[2-Fluoro-5-[(4-methyl-1-piperidyl)sulfonyl]phenyl]boronic acid; 2-Fluoro-5-((4-methylpiperidin-1-yl)sulfonyl)benzeneboronic acid; Boronic acid, B-[2-fluoro-5-[(4-methyl-1-piperidinyl)sulfonyl]phenyl]-; (2-Fluoro-5-(4-methylpiperidine-1-sulfonyl)phenyl)boronic acid; CAS 1704097-14-2; 1704097-14-2
EINECS	Contact for details

Quality Control

Our (2-Fluoro-5-((4-Methylpiperidin-1-yl)sulfonyl)phenyl)boronic acid is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing, including HPLC for purity and NMR for structural confirmation, to ensure it meets the high standards required for sensitive cross-coupling applications. A comprehensive Certificate of Analysis (COA) detailing identity, purity, and impurity profiles is provided with every shipment.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at a controlled room temperature (15-25°C). This compound is hygroscopic (moisture-sensitive) and should be handled under an inert atmosphere (e.g., nitrogen or argon) for long-term storage and when dispensing to prevent degradation.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to structure
Identification (NMR)	Conforms to structure
Purity (HPLC)	≥ 95%
Water Content (KF)	≤ 1.0%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.