Description

(4-Fluoro-3-Morpholinophenyl)Boronic Acid is a high-value boronic acid derivative featuring a morpholine and fluorine substituent on the aromatic ring. This compound is a critical building block in modern synthetic chemistry, enabling the formation of carbon-carbon bonds via the versatile Suzuki-Miyaura cross-coupling reaction. It is primarily utilized by research institutions and pharmaceutical companies engaged in the development of novel active pharmaceutical ingredients (APIs), agrochemicals, and advanced materials.

Application

• Pharmaceutical Intermediate: A key precursor in the synthesis of complex drug candidates, particularly those targeting central nervous system (CNS) disorders and oncology.
• Agrochemical Research: Used to construct novel heterocyclic compounds for the development of new pesticides and herbicides with enhanced efficacy.
• Material Science: Serves as a monomer or cross-linking agent in the creation of advanced polymers, liquid crystals, and organic electronic materials.
• Chemical Synthesis: Enables the efficient, palladium-catalyzed introduction of the (4-fluoro-3-morpholinophenyl) moiety into complex molecular architectures.
• Library Synthesis: Employed in high-throughput and combinatorial chemistry for generating diverse compound libraries for biological screening.
• Ligand & Catalyst Development: Used to prepare novel bidentate or tridentate ligands for catalysis and metal-organic frameworks (MOFs).

Basic Information

Product Name	(4-Fluoro-3-Morpholinophenyl)Boronic Acid
CAS No.	1704073-35-7
Molecular Formula	C10H13BFNO3
Molecular Weight	225.03 g/mol
Synonyms	(4-Fluoro-3-morpholin-4-ylphenyl)boronic acid; (4-Fluoro-3-morpholinophenyl)boronic acid; 3-Morpholino-4-fluorophenylboronic acid; 4-Fluoro-3-morpholinobenzeneboronic acid; B-(4-Fluoro-3-morpholinophenyl)boronic acid; Boronic acid, B-(4-fluoro-3-morpholinophenyl)-; 1704073-35-7; 4-Fluoro-3-morpholinophenylboronic Acid
EINECS	Contact for details

Quality Control

Our (4-Fluoro-3-Morpholinophenyl)Boronic Acid is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing, including HPLC, NMR, and elemental analysis, to ensure high purity and batch-to-batch consistency. Certificates of Analysis (COA) detailing all specifications are provided to guarantee compliance with your research and development requirements.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at a controlled room temperature (15-25°C). Due to its hygroscopic (moisture-sensitive) nature, the container must be kept tightly sealed under an inert atmosphere (e.g., nitrogen or argon) after opening to prevent degradation.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (IR)	Conforms to structure
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 1.0%
Heavy Metals	≤ 20 ppm
Residue on Ignition	≤ 0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.