Description

4-Fluoro-2-((2-Methoxyethoxy)Methyl)Phenylboronic Acid is a sophisticated organoboron compound designed for advanced synthetic chemistry. This boronic acid derivative is a critical building block in modern cross-coupling reactions, enabling the precise construction of complex molecular architectures. It is primarily utilized by research chemists and process development scientists in the pharmaceutical and agrochemical industries for the synthesis of novel active ingredients and functional materials.

Application

• Suzuki-Miyaura Cross-Coupling Reactions: A key reagent for forming carbon-carbon bonds between aryl halides and this boronic acid, essential for creating biaryl structures in drug discovery.
• Pharmaceutical Intermediate Synthesis: Serves as a versatile precursor in the multi-step synthesis of potential active pharmaceutical ingredients (APIs), especially those requiring a fluorinated aromatic moiety.
• Agrochemical Research: Used in the development of new herbicides, fungicides, and insecticides where the specific substitution pattern can influence biological activity and environmental stability.
• Material Science & OLED Development: Employed in the synthesis of organic semiconductors, liquid crystals, and light-emitting materials for electronic devices.
• Chemical Biology & Probe Development: Useful for creating tagged molecules or bioconjugates for studying biological processes, leveraging the boronic acid group's reactivity.
• Process Chemistry & Scale-up: Provides a reliable and high-purity starting point for optimizing synthetic routes from laboratory to pilot plant and commercial production scales.

Basic Information

Product Name	4-Fluoro-2-((2-Methoxyethoxy)Methyl)Phenylboronic Acid
CAS No.	1704065-53-1
Molecular Formula	C10H14BFO4
Molecular Weight	228.03 g/mol
Synonyms	[4-Fluoro-2-[(2-methoxyethoxy)methyl]phenyl]boronic acid; 2-[(2-Methoxyethoxy)methyl]-4-fluorobenzeneboronic acid; 4-Fluoro-2-((2-methoxyethoxy)methyl)benzeneboronic acid; (4-Fluoro-2-((2-methoxyethoxy)methyl)phenyl)boronic acid; 1704065-53-1; 4-Fluoro-2-[(2-methoxyethoxy)methyl]phenylboronic acid
EINECS	Contact for details

Quality Control

Our 4-Fluoro-2-((2-Methoxyethoxy)Methyl)Phenylboronic Acid is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing to ensure high purity and consistency, meeting the stringent requirements for research and process chemistry. Certificates of Analysis (COA) detailing purity, identity, and impurity profiles are available for every lot upon request.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at room temperature (15-25°C). This compound is hygroscopic (moisture-sensitive) and should be handled under an inert atmosphere (e.g., nitrogen or argon) when possible to prevent degradation.

Specification

Item	Specification
Appearance	White to off-white powder or crystalline solid
Identification (IR)	Conforms to structure
Purity (HPLC)	≥95% (Typical 97-99%)
Water Content (KF)	≤1.0%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.