Description

(2-Fluoro-4-((4-Hydroxypiperidin-1-Yl)Methyl)Phenyl)Boronic Acid is a sophisticated boronic acid derivative and a key advanced pharmaceutical intermediate (API) in modern synthetic chemistry. Its core value lies in its dual functionality, serving as a crucial building block in the synthesis of complex molecules via Suzuki-Miyaura cross-coupling reactions. This compound is essential for research and development chemists in the pharmaceutical and agrochemical industries, particularly for creating novel drug candidates and active ingredients.

Application

• Pharmaceutical Intermediate: A critical precursor in the synthesis of active pharmaceutical ingredients (APIs) for oncology, neurology, and other therapeutic areas.
• Suzuki-Miyaura Cross-Coupling Reagent: Enables the formation of carbon-carbon bonds to construct complex biaryl structures, a cornerstone of modern medicinal chemistry.
• Agrochemical Research: Used in the development of new herbicides, fungicides, and insecticides with enhanced efficacy.
• Material Science: Serves as a monomer or building block for creating novel organic electronic materials and polymers.
• Chemical Biology & Probe Development: Utilized in the design of molecular probes and sensors for biological target identification and validation.
• Process Chemistry & Scale-up: Supports route scouting and optimization for the commercial-scale manufacturing of fine chemicals.

Basic Information

Product Name	(2-Fluoro-4-((4-Hydroxypiperidin-1-Yl)Methyl)Phenyl)Boronic Acid
CAS No.	1704064-23-2
Molecular Formula	C12H17BFNO3
Molecular Weight	253.08 g/mol
Synonyms	[2-Fluoro-4-[(4-hydroxypiperidin-1-yl)methyl]phenyl]boronic acid; 1-[(3-Fluoro-4-boronophenyl)methyl]-4-piperidinol; (2-Fluoro-4-((4-Hydroxy-1-piperidinyl)Methyl)Phenyl)Boronic Acid; Boronic acid, B-[2-fluoro-4-[(4-hydroxy-1-piperidinyl)methyl]phenyl]-; 1704064-23-2; 4-(4-Hydroxypiperidin-1-ylmethyl)-2-fluorophenylboronic acid; 2-Fluoro-4-((4-hydroxypiperidin-1-yl)methyl)benzeneboronic acid
EINECS	Contact for details

Quality Control

Our (2-Fluoro-4-((4-Hydroxypiperidin-1-Yl)Methyl)Phenyl)Boronic Acid is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing, including HPLC, NMR, and mass spectrometry, to ensure high purity and batch-to-batch consistency. Certificates of Analysis (COA) detailing all specifications are provided with every shipment to support your quality assurance and regulatory compliance needs.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at a controlled room temperature (15-25°C). This compound is hygroscopic (moisture-sensitive) and should be handled under an inert atmosphere (e.g., nitrogen or argon) when possible to maintain stability and purity. Keep away from incompatible materials.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to structure
Identification (NMR)	Conforms to structure
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 1.0%
Residue on Ignition	≤ 0.5%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.