Description

2-Fluoro-4-(4-Morpholinylcarbonyl)Benzeneboronic Acid, 97% is a high-purity boronic acid derivative featuring a morpholine carbonyl substituent, serving as a critical building block in modern synthetic chemistry. Its value lies in enabling precise carbon-carbon bond formation via Suzuki-Miyaura cross-coupling reactions, a cornerstone for constructing complex molecular architectures. This compound is essential for researchers and process chemists in the pharmaceutical, agrochemical, and advanced materials sectors who require reliable, high-quality intermediates for drug discovery and specialty chemical synthesis.

Application

• Pharmaceutical Intermediate: Key precursor in the synthesis of active pharmaceutical ingredients (APIs) and drug candidates, particularly for kinase inhibitors and other small molecule therapeutics.
• Agrochemical Synthesis: Used in the research and development of novel herbicides, fungicides, and insecticides requiring specific fluorinated aromatic structures.
• Material Science: Building block for creating functionalized polymers, liquid crystals, and organic electronic materials through palladium-catalyzed coupling.
• Chemical Research & Development: A versatile reagent in academic and industrial R&D labs for exploring new synthetic pathways and creating compound libraries.
• Suzuki-Miyaura Cross-Coupling: The primary application is as a boron-containing coupling partner with aryl/vinyl halides or triflates to form biaryl and other conjugated systems.
• Ligand and Catalyst Development: Potential use in the synthesis of novel ligands for catalysis or as a component in metal-organic frameworks (MOFs).

Basic Information

Item	Detail
Product Name	2-Fluoro-4-(4-Morpholinylcarbonyl)Benzeneboronic Acid, 97%
CAS No.	1092500-69-0
Molecular Formula	C11H13BFNO4
Molecular Weight	265.04 g/mol
Synonyms	(2-Fluoro-4-(morpholine-4-carbonyl)phenyl)boronic acid; 2-Fluoro-4-(morpholine-4-carbonyl)benzeneboronic acid; 4-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)-3-fluorobenzoic acid morpholide; 2-Fluoro-4-morpholinocarbonylbenzeneboronic acid; Boronic acid, B-[2-fluoro-4-(4-morpholinylcarbonyl)phenyl]-; [2-Fluoro-4-(morpholine-4-carbonyl)phenyl]boronic acid
EINECS	Contact for details

Quality Control

Our 2-Fluoro-4-(4-Morpholinylcarbonyl)Benzeneboronic Acid, 97% is manufactured under strict quality management systems. Every batch undergoes rigorous analytical testing, including HPLC for purity and identity confirmation by NMR and IR spectroscopy, to ensure it meets the specified 97% minimum purity. Certificates of Analysis (COA) with full traceability are available upon request.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at room temperature (15-25°C). This material is hygroscopic (moisture-sensitive) and should be handled under a dry inert atmosphere (e.g., nitrogen or argon) when opening to prevent degradation.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to structure
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 1.0%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.