Description

[1,3'-Biazetidine]-1'-Carboxylic Acid,3-Amino-, 1,1-Dimethylethyl Ester is a high-purity, protected amino acid derivative featuring a unique biazetidine scaffold. This compound is a critical pharmaceutical intermediate and building block for advanced medicinal chemistry research, enabling the synthesis of novel bioactive molecules. It is primarily utilized by R&D chemists and process development scientists in the pharmaceutical, biotechnology, and agrochemical industries for the development of new therapeutic agents and fine chemicals.

Application

• Pharmaceutical Intermediate: A key building block for the synthesis of novel drug candidates, particularly those targeting protease inhibition or requiring constrained peptide mimetics.
• Peptidomimetic Research: Used to construct complex, conformationally restricted peptide analogs to enhance metabolic stability and receptor selectivity.
• Chemical Biology Probes: Serves as a scaffold for developing activity-based probes and molecular tools to study enzyme function and biological pathways.
• Agrochemical Synthesis: Potential intermediate in the development of new generation herbicides or fungicides with novel modes of action.
• Material Science: Exploration as a monomer or cross-linking agent for specialty polymers with unique thermal or mechanical properties.
• Academic & Contract Research: Fundamental research in organic methodology and heterocyclic chemistry within university and CRO laboratories.

Basic Information

Product Name	[1,3'-Biazetidine]-1'-Carboxylic Acid,3-Amino-, 1,1-Dimethylethyl Ester
CAS No.	1026796-77-9
Molecular Formula	C11H21N3O2
Molecular Weight	227.30 g/mol
Synonyms	tert-Butyl 3-amino[1,3']biazetidinyl-1'-carboxylate; 1,1-Dimethylethyl 3-amino-1,3'-biazetidine-1'-carboxylate; Boc-3-amino[1,3']biazetidine; 3-Amino[1,3']biazetidinyl-1'-carboxylic acid tert-butyl ester; N-Boc-3-amino-1,3'-biazetidine; (3-Amino[1,3']biazetidin-1'-yl)-tert-butoxycarbonyl; Biazetidine amino acid Boc ester
EINECS	Contact for details

Quality Control

Our [1,3'-Biazetidine]-1'-Carboxylic Acid,3-Amino-, 1,1-Dimethylethyl Ester is manufactured under strict quality control protocols to ensure batch-to-batch consistency and high purity. Production adheres to cGMP guidelines where applicable. Each lot is accompanied by a comprehensive Certificate of Analysis (COA) detailing identity, purity, and impurity profiles, available upon request. We are committed to meeting the stringent requirements of pharmaceutical R&D and scale-up processes.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at a controlled room temperature (15-25°C). This compound is hygroscopic (moisture-sensitive) and should be handled under anhydrous conditions to maintain stability and purity. For long-term storage, consider storing under an inert atmosphere.

Specification

Item	Specification
Appearance	White to off-white solid
Identification (IR)	Conforms to structure
Identification (NMR)	Conforms to structure
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 0.5%
Residual Solvents (GC)	Meets ICH guidelines

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.