Description

Tianeptine Metabolite Mc5 Sodium Salt is a key reference standard and active pharmaceutical ingredient (API) intermediate, specifically the sodium salt of a major metabolite of the antidepressant tianeptine. This compound is critical for pharmaceutical research and development, enabling precise pharmacokinetic studies, metabolic pathway analysis, and the development of improved therapeutic agents. It is primarily utilized by research institutions, analytical laboratories, and pharmaceutical companies engaged in neuroscience, drug metabolism studies, and quality control for related pharmaceutical products.

Application

• Pharmaceutical Reference Standard: Used as a certified standard for the quantitative and qualitative analysis of tianeptine and its metabolites in biological matrices and pharmaceutical formulations.
• Metabolite Research: Essential for studying the pharmacokinetics, bioavailability, and metabolic pathways of tianeptine in preclinical and clinical research.
• Active Pharmaceutical Ingredient (API) Intermediate: Serves as a high-purity building block in the synthesis and development of novel pharmaceutical compounds targeting the central nervous system.
• Analytical Method Development: Employed to develop and validate sensitive analytical methods, such as HPLC and LC-MS/MS, for drug monitoring and impurity profiling.
• Neuroscience & Neuropsychopharmacology Research: Used in vitro and in vivo studies to investigate the mechanisms of action and effects of tianeptine metabolites.
• Quality Control & Assurance: Critical for ensuring the purity, identity, and consistency of tianeptine-based drug substances and products in GMP environments.

Basic Information

Product Name	Tianeptine Metabolite Mc5 Sodium Salt
CAS No.	115220-11-6
Molecular Formula	Contact for details
Molecular Weight	Contact for details
Synonyms	MC5 Sodium Salt; Tianeptine Acid Metabolite Sodium Salt; 7-[(3-chloro-6-methyl-5,5-dioxido-6,11-dihydrodibenzo[c,f][1,2]thiazepin-11-yl)amino]heptanoic acid sodium salt; Sodium 7-[(3-chloro-6,11-dihydro-6-methyl-5,5-dioxodibenzo[c,f][1,2]thiazepin-11-yl)amino]heptanoate; Tianeptine Metabolite (Acid) Sodium Salt
EINECS	Contact for details

Quality Control

Our Tianeptine Metabolite Mc5 Sodium Salt is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing to ensure high purity and consistency, meeting the stringent requirements for pharmaceutical reference standards and API intermediates. A comprehensive Certificate of Analysis (COA) detailing identity, purity, and impurity profiles by methods such as HPLC, NMR, and MS is provided with every shipment to support your research and regulatory needs.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at controlled room temperature (15-25°C). Due to its hygroscopic (moisture-sensitive) nature, the container must be kept tightly sealed in a dry environment to prevent degradation. For long-term storage, consider desiccants or inert atmosphere.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (HPLC)	Conforms to reference standard
Identification (NMR)	Conforms to structure
Assay (HPLC)	≥ 98.0%
Related Substances (HPLC)	Total impurities ≤ 2.0%
Water Content (KF)	≤ 5.0%
Residual Solvents (GC)	Complies with ICH guidelines

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.