Tinib Antineoplastic Drugs

Tinib Antineoplastic Drugs

Tinib antineoplastic drugs are a major class of targeted cancer therapies that inhibit dysregulated tyrosine kinases or serine/threonine kinases involved in tumor growth, angiogenesis, and metastasis. Represented by imatinib, erlotinib, gefitinib, sunitinib, sorafenib, and numerous next-generation inhibitors, these APIs block oncogenic signaling pathways such as EGFR, VEGFR, PDGFR, BCR-ABL, ALK, and RET. Their precision targeting enables high efficacy with reduced systemic toxicity compared to traditional chemotherapy. Tinib drugs are widely used in leukemia, lung cancer, renal cancer, gastrointestinal stromal tumors, and melanoma. Resistance caused by kinase mutations has led to the development of multi-targeted and mutation-specific inhibitors, making tinibs a cornerstone of precision oncology.

n-(3-((2-((3-Fluoro-4-(4-Methylpiperazin-1-Yl)Phenyl)Amino)-7H-Pyrrolo[2,3-D]Pyrimidin-4-Yl)Oxy)Phenyl)Acrylamide Maleate CAS NO 1557268-88-8

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CAS No.:1557268-88-8

Grade:Pharmacy Grade

Content:99.90%

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Bgb-3111 CAS NO 1558036-85-3

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CAS No.:1558036-85-3

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Content:99.90%

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Crenolanib Trifluoroacetic Acid Salt CAS NO 1797008-57-1

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CAS No.:1797008-57-1

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Content:99.90%

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Tyk2-In-5 CAS NO 1797432-62-2

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CAS No.:1797432-62-2

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Content:99.90%

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1-((2R,5S)-5-((7H-Pyrrolo[2,3-D]Pyrimidin-4-Yl)Amino)-2-Methylpiperidin-1-Yl)Prop-2-En-1-One CAS NO 1792180-79-0

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CAS No.:1792180-79-0

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1-((2S,5R)-5-((7H-Pyrrolo[2,3-D]Pyrimidin-4-Yl)Amino)-2-Methylpiperidin-1-Yl)Prop-2-En-1-One CAS NO 1792180-81-4

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CAS No.:1792180-81-4

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Content:99.90%

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Gs-9876 (Lanraplenib) CAS NO 1800046-95-0

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CAS No.:1800046-95-0

Grade:Pharmacy Grade

Content:99.90%

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Lxh254,Lxh-254 CAS NO 1800398-38-2

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CAS No.:1800398-38-2

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Content:99.90%

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