Description

Lavoltidine is a potent and selective histamine H2-receptor antagonist. This compound is of significant interest in pharmaceutical research and development for its potential therapeutic applications. It is primarily utilized by researchers and manufacturers in the pharmaceutical industry for the development of novel treatments targeting gastric acid secretion.

Application

• Pharmaceutical Intermediate: Serves as a key building block in the synthesis of advanced active pharmaceutical ingredients (APIs).
• Gastrointestinal Research: Used in preclinical and clinical research studies investigating new anti-ulcer and acid-suppressing medications.
• Biochemical Tool: Employed as a selective ligand in pharmacological assays to study histamine H2-receptor function and signaling pathways.
• Reference Standard: Acts as a high-purity analytical standard for quality control and method validation in pharmaceutical laboratories.
• Drug Discovery: Integral to medicinal chemistry programs aimed at developing next-generation histamine H2-receptor antagonists with improved profiles.

Basic Information

Product Name	Lavoltidine
CAS No.	76956-02-0
Molecular Formula	C19H21N5O3S
Molecular Weight	399.47 g/mol
Synonyms	Lavoltidine; FRG-8813; FRG 8813; 2-[[[2-[(Aminoiminomethyl)amino]-4-thiazolyl]methyl]thio]-N-(2-fluoroethyl)acetamide; 2-({[2-(Carbamimidamido)-1,3-thiazol-4-yl]methyl}sulfanyl)-N-(2-fluoroethyl)acetamide; FRG8813
EINECS	Contact for details

Quality Control

Our Lavoltidine is manufactured under strict quality management systems. Each batch undergoes comprehensive analytical testing, including HPLC for purity and identity confirmation (IR, NMR), to ensure it meets the high standards required for pharmaceutical research and development. Certificates of Analysis (COA) with detailed specifications are provided and can be tailored to meet specific project requirements.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at controlled room temperature (15-25°C). Due to its hygroscopic nature, the container must be kept tightly sealed in a dry environment to prevent moisture absorption.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to reference spectrum
Identification (HPLC)	Retention time matches reference standard
Assay (HPLC)	≥ 98.0%
Related Substances (HPLC)	Total impurities ≤ 2.0% Any single impurity ≤ 1.0%
Water Content (KF)	≤ 1.0%
Residue on Ignition	≤ 0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.